SCHEMBL19210394

SCHEMBL19210394

COc1ccc(-c2nc(C(CCOc3ccc(F)c(C(N)=O)c3F)C(=O)O)oc2Br)cc1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSA P10619 1/20 0.33
PPARD Q03181 5/20 0.33
TP53 P04637 1/20 0.33
IKBKB O14920 1/20 0.33
TPH1 P17752 4/20 0.33
AKR1C3 P42330 1/20 0.33
AKR1C2 P52895 1/20 0.33
PTGS2 P35354 3/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
PTGS1 P23219 1/20 0.32
PDE3A Q14432 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19210475 0.91 FFAR4 (0.33) CTSA
SCHEMBL19210491 0.90 AKR1C3 (0.38) CTSAPPARDIKBKBAKR1C3AKR1C2
SCHEMBL19210450 0.90 FFAR4 (0.35) PPARD
SCHEMBL19210420 0.88 PTGS2 (0.34) CTSAPTGS2PTGDR2PTGS1
SCHEMBL19210513 0.88 PTPN1 (0.34) PPARDIKBKB
SCHEMBL19210439 0.87 SCN9A (0.34) PTGDR2
SCHEMBL19210396 0.86 S1PR1 (0.35) TP53TPH1
SCHEMBL13734082 0.83 PPARD (0.37) PPARDTP53IKBKBPTGDR2HTT
SCHEMBL19210393 0.82 MAPT (0.35) CTSAPPARDIKBKBPTGS2PTGDR2
SCHEMBL15674929 0.82 IKBKB (0.36) CTSATP53IKBKBPTGDR2PDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2699557-B1 3-(OXAZOL-2-YL-ETHOXY)- AND 3-(THIAZOL-2-YL-ETHOXY)-BENZAMIDE DERIVATIVES AS ANTI-BACTERIAL AGENTS BIOTA SCIENT MANAGEMENT (AU) 2017-08-16 EP claimed