SCHEMBL1921731

SCHEMBL1921731

O=C(O)Oc1ccc2nn(-c3ccccc3)c(Cc3ccccc3)c2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 1/20 0.40
MDM2 Q00987 3/20 0.39
CHEK1 O14757 1/20 0.36
AURKA O14965 1/20 0.36
CSNK1A1 P48729 1/20 0.36
CDK8 P49336 1/20 0.36
NEK2 P51955 1/20 0.36
LIMK1 P53667 1/20 0.36
CDK5 Q00535 1/20 0.36
DYRK1A Q13627 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
HSP90AA1 P07900 1/20 0.35
PLA2G4A P47712 1/20 0.35
MPO P05164 1/20 0.35
BCL2 P10415 2/20 0.35
MCL1 Q07820 2/20 0.35
KMT2A Q03164 2/20 0.35
DPP4 P27487 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921251 0.84 PLA2G2A (0.47) PLA2G2AALDH1A1MPOKMT2AMAPT
SCHEMBL1921689 0.81 IP6K1 (0.48) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL13984695 0.79 NPC1 (0.44) ALDH1A1HSP90AA1MPOMAPTRAB9A
SCHEMBL1920882 0.77 ELANE (0.37) PLA2G2AMDM2CHEK1AURKACSNK1A1
SCHEMBL1921321 0.75 MPO (0.50) ALDH1A1MPOKMT2ARAB9ANPC1
SCHEMBL28748682 0.74 MPO (0.45) PLA2G2AALDH1A1LMNAMPOKMT2A
SCHEMBL1921325 0.73 CCNC (0.42) CDK8ALDH1A1LMNANPSR1
SCHEMBL1921521 0.73 ALDH1A1 (0.44) PLA2G2AALDH1A1LMNAMPOMAPT
SCHEMBL1921363 0.73 CHEK1 (0.50) CHEK1AURKACSNK1A1CDK8NEK2
SCHEMBL1921320 0.72 ALDH1A1 (0.54) ALDH1A1MPOKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170833-B1 A TRANSITION METAL CATALYZED SYNTHESIS OF 2H-INDAZOLES SANOFI AVENTIS (FR) 2011-06-01 EP claimed