SCHEMBL19230370

SCHEMBL19230370

COC(=O)c1ccc2c(c1)CCC(c1ccc(O)nc1C(F)(F)F)O2

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC8A1 P32418 10/20 0.37
HSD11B1 P28845 1/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
NISCH Q9Y2I1 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
HTT P42858 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NOTUM Q6P988 1/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
RBP4 P02753 1/20 0.35
AKR1C3 P42330 1/20 0.34
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230992 0.82 ESR2 (0.44) SLC8A1CHRNB2CHRNA4NOTUMESR1
SCHEMBL19230821 0.80 ESR1 (0.40) SLC8A1ESR1ESR2
SCHEMBL19230824 0.79 NOTUM (0.43) SLC8A1NOTUMRBP4
SCHEMBL19230375 0.79 ESR2 (0.46) SLC8A1CHRNB2CHRNA4NISCHESR1
SCHEMBL19230775 0.78 ESR1 (0.38) SLC8A1HSD11B1ESR1ESR2AKR1C3
SCHEMBL19230993 0.77 ESR1 (0.47) SLC8A1CHRNB2CHRNA4NISCHESR1
SCHEMBL19230656 0.76 ESR1 (0.49) CHRNB2CHRNA4NISCHKDM4EALDH1A1
SCHEMBL19230805 0.76 ESR1 (0.49) CHRNB2CHRNA4NISCHKDM4EALDH1A1
SCHEMBL19230687 0.76 ESR1 (0.46) SLC8A1ESR1ESR2
SCHEMBL19230310 0.76 ESR1 (0.49) CHRNB2CHRNA4NISCHKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed