SCHEMBL19230775

SCHEMBL19230775

N#Cc1ccc2c(c1)CCC(c1ccc(O)nc1C(F)(F)F)O2

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
PTGS2 P35354 1/20 0.33
SLC8A1 P32418 2/20 0.32
HSD11B1 P28845 1/20 0.32
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
AR P10275 4/20 0.31
PNMT P11086 1/20 0.31
FDPS P14324 1/20 0.31
LRRK2 Q5S007 1/20 0.31
AKR1C3 P42330 1/20 0.31
TRPV1 Q8NER1 1/20 0.30
P2RY6 Q15077 1/20 0.30
PGR P06401 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230821 0.84 ESR1 (0.40) ESR1ESR2SLC8A1AR
SCHEMBL19230370 0.78 SLC8A1 (0.37) ESR1ESR2SLC8A1HSD11B1AKR1C3
SCHEMBL19230545 0.74 ESR1 (0.53) ESR1ESR2CYP11B2
SCHEMBL11048933 0.71 ESR1 (0.57) ESR1ESR2SLC8A1PNMT
SCHEMBL3488386 0.67 ESR1 (0.56) ESR1ESR2SLC8A1PNMT
SCHEMBL19230671 0.65 ESR2 (0.50) ESR1ESR2CYP11B2
SCHEMBL24101932 0.65 DPP4 (0.41) CYP11B1CYP11B2PGR
SCHEMBL10509432 0.65 DRD2 (0.36) ESR1ESR2PNMT
SCHEMBL10510220 0.64 DRD2 (0.37) ESR1ESR2PTGS2CYP11B1CYP11B2
SCHEMBL1029126 0.63 PGR (0.56) CYP11B1CYP11B2PNMTLRRK2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed