SCHEMBL19230656

SCHEMBL19230656

COC(=O)c1ccc2c(c1)CC[C@H](c1ccc(O)cc1Cl)O2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.49
ESR2 Q92731 5/20 0.49
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
RAB9A P51151 2/20 0.38
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230805 1.00 ESR1 (0.49) ESR1ESR2SLC6A2SLC6A4SLC6A3
SCHEMBL19230310 1.00 ESR1 (0.49) ESR1ESR2SLC6A2SLC6A4SLC6A3
SCHEMBL19230672 0.91 ESR2 (0.46) ESR1ESR2SLC6A2SLC6A4SLC6A3
SCHEMBL19230647 0.89 RAB9A (0.43) SLC6A2SLC6A4SLC6A3RAB9ACA12
SCHEMBL19230993 0.88 ESR1 (0.47) ESR1ESR2RAB9APDK1PDK2
SCHEMBL19230375 0.87 ESR2 (0.46) ESR1ESR2RAB9APDK1PDK2
SCHEMBL19230623 0.87 ESR1 (0.45) ESR1ESR2SLC6A2SLC6A4SLC6A3
SCHEMBL28649906 0.86 ESR1 (0.53) ESR1ESR2PDK1PDK2PDK3
SCHEMBL19230992 0.84 ESR2 (0.44) ESR1ESR2RAB9APDK1PDK2
SCHEMBL19230616 0.83 ESR2 (0.65) ESR1ESR2RAB9ACA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed