SCHEMBL19230593

SCHEMBL19230593

COC(=O)c1cccc2c1CCC(c1ccc(OC)cc1Cl)O2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44
TAS1R2 Q8TE23 1/20 0.44
DRD2 P14416 2/20 0.41
DRD4 P21917 2/20 0.41
DRD1 P21728 1/20 0.41
DRD5 P21918 1/20 0.41
DRD3 P35462 1/20 0.39
HTR5A P47898 1/20 0.39
DPP4 P27487 3/20 0.38
CYP19A1 P11511 2/20 0.38
TSHR P16473 1/20 0.37
CHRM2 P08172 2/20 0.36
CHRM4 P08173 2/20 0.36
CHRM5 P08912 2/20 0.36
CHRM1 P11229 2/20 0.36
CHRM3 P20309 2/20 0.36
MCOLN1 Q9GZU1 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19230591 0.88 DRD2 (0.43) TAS1R3TAS1R1TAS1R2DRD2DRD4
SCHEMBL19230525 0.83 TAS1R3 (0.46) TAS1R3TAS1R1TAS1R2DRD2DRD4
SCHEMBL19230749 0.80 TAS1R3 (0.33) TAS1R3TAS1R1TAS1R2DRD2DRD4
SCHEMBL19230747 0.78 NR1H4 (0.56)
SCHEMBL19230597 0.77 DRD2 (0.43) DRD2DRD4DRD1DRD5DRD3
SCHEMBL27317222 0.73 DRD2 (0.44) DRD2DRD4DRD3HTR5ATSHR
SCHEMBL19538256 0.72 DPP4 (0.64) DPP4
SCHEMBL19230604 0.71 DRD2 (0.39) TAS1R3TAS1R1TAS1R2DRD2DRD4
SCHEMBL19313488 0.70 DPP4 (0.65) DPP4TSHRKDM4EALDH1A1HSD17B10
SCHEMBL1180038 0.67 TYK2 (0.57) KDM4ECYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108602811-B FXR receptor agonists 轩竹生物科技有限公司 2021-11-16 CN disclosed
WO-2017133521-A1 FXR RECEPTOR AGONIST 山东轩竹医药科技有限公司 2017-08-10 WO disclosed