SCHEMBL19230910

SCHEMBL19230910

Cn1nc(I)c2cc(F)cnc21

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SPR P35270 3/20 0.36
GSK3B P49841 1/20 0.36
ALDH1A1 P00352 1/20 0.31
PDE10A Q9Y233 1/20 0.31
POLB P06746 1/20 0.31
HTR3A P46098 1/20 0.31
MAP3K14 Q99558 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16167735 0.80 SPR (0.52) SPRGSK3BPDE10APOLB
SCHEMBL12703712 0.79 HSD17B10 (0.46) SPRGSK3BALDH1A1POLB
SCHEMBL16199065 0.79 HPGD (0.46) SPRGSK3BALDH1A1POLB
SCHEMBL3026539 0.79 GSK3B (0.43) SPRGSK3BALDH1A1POLB
SCHEMBL19480629 0.79 GSK3B (0.58) SPRGSK3BALDH1A1PDE10APOLB
SCHEMBL25527223 0.76 GSK3B (0.38) SPRGSK3BPDE10APOLBHTR3A
SCHEMBL24331224 0.71 BRD4 (0.50) GSK3BHTR3A
SCHEMBL14488171 0.70 GRIN1 (0.37)
SCHEMBL19230912 0.70 ADORA2A (0.32) ALDH1A1PDE10A
SCHEMBL3034786 0.69 SPR (0.33) SPRGSK3BPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170233413-A1 SUBSTITUTED ANNULATED PYRIMIDINES AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2017-08-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170233413-A1 SUBSTITUTED ANNULATED PYRIMIDINES AND USE THEREOF TYMP, DPYD, TYMS SPR 1342/4885GSK3B 4414/4885ALDH1A1 660/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.