SCHEMBL1923323

SCHEMBL1923323

O=C(CC1CC1)N[C@H]1CC[C@H](CCN2CCC(C(=O)c3ccc(F)cc3Cl)CC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 15/20 0.50
DRD3 P35462 15/20 0.50
HPGD P15428 1/20 0.48
DRD2 P14416 6/20 0.47
ACKR3 P25106 1/20 0.45
HSD11B1 P28845 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL228867 1.00 HTR2A (0.50) HTR2ADRD3HPGDDRD2ACKR3
SCHEMBL228147 0.89 ACKR3 (0.54) HTR2ADRD3HPGDDRD2ACKR3
SCHEMBL228146 0.89 ACKR3 (0.54) HTR2ADRD3HPGDDRD2ACKR3
SCHEMBL230475 0.87 DRD3 (0.60) HTR2ADRD3DRD2
SCHEMBL225949 0.86 HSD11B1 (0.47) HTR2ADRD3DRD2ACKR3HSD11B1
SCHEMBL228931 0.86 DRD2 (0.59) HTR2ADRD3HPGDDRD2
SCHEMBL229290 0.85 DRD3 (0.61) HTR2ADRD3DRD2ACKR3
SCHEMBL227883 0.84 ACKR3 (0.45) HTR2ADRD3DRD2ACKR3
SCHEMBL230816 0.84 HSD11B1 (0.49) HTR2ADRD2ACKR3HSD11B1
SCHEMBL27758351 0.84 HSD11B1 (0.49) HTR2ADRD2ACKR3HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185513-B1 BENZOYL-PIPERIDINE DERIVATIVES AS DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2011-06-08 EP claimed