SCHEMBL19236012

SCHEMBL19236012

CCN(C(=O)OC(C)(C)C)/C(=N\C(=O)OC(C)(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA7 P43166 1/20 0.34
CA14 Q9ULX7 1/20 0.34
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
CTSK P43235 1/20 0.31
PTGES O14684 1/20 0.31
TDP1 Q9NUW8 1/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3444153 0.82 CA14 (0.31) CA12CA1CA7CA14TDP1
SCHEMBL24669520 0.82 CA1 (0.36) CA12CA1CA7CA14KDM4E
SCHEMBL22651785 0.80 CTSK (0.33) CA1CA7CTSKPTGESKMT2A
SCHEMBL7038864 0.80 CA12 (0.30) CA12CA1CA7CA14PTGES
SCHEMBL16808277 0.80 CA12 (0.30) CA12CA1CA7CA14PTGES
SCHEMBL8193600 0.78 CTSK (0.33) CA12CA1CA7CA14CTSK
SCHEMBL19465020 0.78 CTSK (0.33) CA12CA1CA7CA14CTSK
SCHEMBL8193597 0.78 CTSK (0.33) CA12CA1CA7CA14CTSK
SCHEMBL18296719 0.78 TDP1 (0.40) CA12CA1CA14TDP1KMT2A
SCHEMBL20207093 0.78 TDP1 (0.40) CA12CA1CA14TDP1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170233335-A1 INHIBITORS OF HIV-1 ENTRY AND METHODS OF USE THEREOF BRYN MAWR COLLEGE 2017-08-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170233335-A1 INHIBITORS OF HIV-1 ENTRY AND METHODS OF USE THEREOF CD4, CD81, ICAM1 CA12 3447/4885CA1 3298/4885CA7 4351/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.