SCHEMBL8193597

SCHEMBL8193597

CN(C)/C(=N\C(=O)OC(C)(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.33
CA1 P00915 2/20 0.33
CA7 P43166 2/20 0.33
CA12 O43570 1/20 0.33
CA14 Q9ULX7 1/20 0.33
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
PTGES O14684 1/20 0.32
CA2 P00918 1/20 0.31
DGAT1 O75907 1/20 0.31
MIF P14174 1/20 0.30
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19465020 1.00 CTSK (0.33) CTSKCA1CA7CA12CA14
SCHEMBL8193600 1.00 CTSK (0.33) CTSKCA1CA7CA12CA14
SCHEMBL24670538 0.86 CA12 (0.31) CA1CA7CA12CA14NFKB1
SCHEMBL7038864 0.85 CA12 (0.30) CA1CA7CA12CA14PTGES
SCHEMBL16808277 0.85 CA12 (0.30) CA1CA7CA12CA14PTGES
SCHEMBL19460142 0.83 CA12 (0.35) CTSKCA1CA7CA12CA14
SCHEMBL24669520 0.83 CA1 (0.36) CTSKCA1CA7CA12CA14
SCHEMBL3216144 0.83 DGAT1 (0.32) CA1CA7CA12CA14NFKB1
SCHEMBL22730755 0.81 CA12 (0.43) CTSKCA1CA7CA12CA14
SCHEMBL18121932 0.81 CA12 (0.31) CTSKCA1CA7CA12CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100260-A ((3-(1-(2-FLUORO-BIPHENYL-4-YL)-ETHYL)-ISOXAZOL-5-YLIMINO) -MORPHOLIN-4-YL-M ETHYL)-AMINE, FOR EXAMPLE; ADMINISTERING TO TREAT AUTOIMMUNE DISEASES AND INFLAMMATION SUMITOMO PHARMACEUTICAL COMPANY, LIMITED (JP) 2000-08-08 US disclosed