SCHEMBL19250267

SCHEMBL19250267

O=C1COc2ccc(N(C(=O)O)C3CCCCC3)nc2N1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 9/20 0.39
PDE3B Q13370 1/20 0.38
PDE3A Q14432 1/20 0.38
NR3C1 P04150 1/20 0.37
TP53 P04637 2/20 0.35
MEN1 O00255 1/20 0.35
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35
KMT2A Q03164 1/20 0.35
MGLL Q99685 1/20 0.35
KCNH2 Q12809 3/20 0.35
GAA P10253 1/20 0.35
PARP1 P09874 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19250443 0.82 NR3C2 (0.43) NR3C2PDE3BPDE3ANR3C1TP53
SCHEMBL19250277 0.80 NR3C2 (0.39) NR3C2PDE3BPDE3ANR3C1KCNH2
SCHEMBL19629922 0.79 NR3C2 (0.41) NR3C2NR3C1PKMKMT2AMGLL
SCHEMBL19629923 0.78 NR3C2 (0.43) NR3C2NR3C1PKMKCNH2GAA
SCHEMBL19629924 0.78 NR3C2 (0.40) NR3C2NR3C1PKMKMT2AKCNH2
SCHEMBL7977817 0.78 NR3C2 (0.40) NR3C2NR3C1PKMKMT2AGAA
SCHEMBL23871692 0.73 MAPK14 (0.40) NR3C2NR3C1MGLLKCNH2
SCHEMBL23871561 0.71 NR3C2 (0.38) NR3C2NR3C1MGLLKCNH2
SCHEMBL619718 0.70 NR3C2 (0.44) NR3C2NR3C1PKMKMT2AMGLL
SCHEMBL17956629 0.69 NR3C2 (0.37) NR3C2NR3C1TP53MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017137744-A1 HETEROCYCLIC COMPOUNDS, IN PARTICULAR 2-OXO-4,4,5,5,6,6,7,7-OCTAHYDROBENZOXAZOLE DERIVATIVES, AND THEIR USE AS ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2017-08-17 WO disclosed