SCHEMBL19251214

SCHEMBL19251214

CCC(C)(CC)c1cncc(C#N)c1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 3/20 0.37
RAF1 P04049 1/20 0.36
CYP19A1 P11511 1/20 0.35
CYP11B1 P15538 2/20 0.34
PTGER4 P35408 1/20 0.33
CYP1A2 P05177 1/20 0.33
METAP2 P50579 1/20 0.33
USP7 Q93009 2/20 0.33
GRIN1 Q05586 3/20 0.32
GRIN2B Q13224 3/20 0.32
KIF11 P52732 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18935594 0.86 CYP11B2 (0.40) CYP11B2RAF1CYP19A1CYP11B1PTGER4
SCHEMBL19592946 0.82 CNR2 (0.38) CYP11B2RAF1CYP11B1CYP1A2METAP2
SCHEMBL9967844 0.81 KIF11 (0.44) CYP11B2RAF1CYP19A1CYP11B1CYP1A2
SCHEMBL19251665 0.79 CYP11B2 (0.39) CYP11B2RAF1CYP11B1PTGER4CYP1A2
SCHEMBL14822598 0.78 CYP11B2 (0.55) CYP11B2RAF1CYP11B1
SCHEMBL22338688 0.78 CYP1A2 (0.40) CYP11B2RAF1CYP11B1CYP1A2METAP2
SCHEMBL22303444 0.75 CYP11B2 (0.41) CYP11B2RAF1CYP11B1CYP1A2METAP2
SCHEMBL14809739 0.75 CYP11B2 (0.37) CYP11B2RAF1CYP19A1CYP11B1CYP1A2
SCHEMBL2749165 0.73 CYP1A2 (0.49) CYP11B2CYP11B1CYP1A2METAP2GRIN1
SCHEMBL30133235 0.73 CYP1A2 (0.49) CYP11B2CYP11B1CYP1A2METAP2GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed