SCHEMBL19251271

SCHEMBL19251271

CCc1ccc(C(C)N2CCN(CC)CC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.48
MC4R P32245 2/20 0.43
ALDH1A1 P00352 2/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
OGA O60502 1/20 0.42
CHRM2 P08172 3/20 0.42
CHRM1 P11229 2/20 0.42
SIGMAR1 Q99720 2/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CHRM3 P20309 1/20 0.40
DRD3 P35462 1/20 0.40
OPRD1 P41143 1/20 0.40
KCNH2 Q12809 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
TSHR P16473 2/20 0.40
RORC P51449 1/20 0.39
MAPK1 P28482 1/20 0.39
ATM Q13315 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14924035 0.86 CYP2D6 (0.52) CYP2D6MC4RALDH1A1HDAC4HDAC1
SCHEMBL14924473 0.84 ALDH1A1 (0.53) CYP2D6MC4RALDH1A1CHRM2CHRM1
SCHEMBL18403967 0.84 ALDH1A1 (0.53) CYP2D6MC4RALDH1A1CHRM2CHRM1
SCHEMBL12845564 0.84 CYP2D6 (0.48) CYP2D6MC4ROGACHRM2CHRM1
SCHEMBL10112423 0.83 CYP2D6 (0.50) CYP2D6MC4RHDAC4HDAC1CHRM2
SCHEMBL18403964 0.83 GAA (0.54) CYP2D6MC4RALDH1A1HDAC4HDAC1
SCHEMBL14600336 0.82 CYP2D6 (0.74) CYP2D6MC4RALDH1A1HDAC4HDAC1
SCHEMBL20012737 0.82 CYP2D6 (0.74) CYP2D6MC4RALDH1A1HDAC4HDAC1
SCHEMBL10259631 0.79 LTA4H (0.47) CYP2D6MC4RALDH1A1OGATSHR
SCHEMBL24129459 0.79 CYP2D6 (0.44) CYP2D6MC4RALDH1A1CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE46511-E1 Fused pyrimidine derivatives for inhibition of tyrosine kinase activity HANMI SCIENCE CO., LTD. (KR) 2017-08-15 US disclosed