SCHEMBL19251530

SCHEMBL19251530

CCCCC(C)(C)c1ccc2c(c1)C(=O)NC21CC1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 19/20 0.41
CNR1 P21554 18/20 0.41
NPC1 O15118 1/20 0.34
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
CASP3 P42574 1/20 0.34
RAB9A P51151 1/20 0.34
ATM Q13315 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SENP8 Q96LD8 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
SENP6 Q9GZR1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12459166 0.81 ALDH1A1 (0.41) NPC1CASP3RAB9ASENP8SENP7
SCHEMBL23271199 0.68 TDP2 (0.42) SMN1; SMN2
SCHEMBL29683177 0.68 TDP2 (0.42) SMN1; SMN2
SCHEMBL16006554 0.67 PBRM1 (0.42) LMNA
SCHEMBL14992095 0.67 PARP1 (0.45)
SCHEMBL29226241 0.67 TGM2 (0.49)
SCHEMBL30900443 0.67 TGM2 (0.49)
SCHEMBL30095473 0.67 CA9 (0.39) NPC1LMNAMAPK1RAB9ASMN1; SMN2
SCHEMBL17695142 0.66 HPGD (0.57) LMNA
SCHEMBL18410997 0.64 CNR2 (0.43) CNR2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9732083-B2 Tricyclic gyrase inhibitors MERCK SHARP & DOHME CORP. (US) 2017-08-15 US disclosed