SCHEMBL19255037

SCHEMBL19255037

CN(C)[S+]([O-])c1cccc(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
MAPK1 P28482 1/20 0.40
TAAR1 Q96RJ0 3/20 0.39
PYCR1 P32322 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
KDM1A O60341 2/20 0.32
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
C1S P09871 1/20 0.31
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14434282 0.78 ACHE (0.44) ALDH1A1MAPK1TAAR1PARP1
SCHEMBL513922 0.77 ALDH1A1 (0.44) ALDH1A1MAPK1TAAR1KDM1AC1S
SCHEMBL3667921 0.76 ALDH1A1 (0.42) ALDH1A1MAPK1TAAR1KDM1AC1S
SCHEMBL18933061 0.74 CYP2A6 (0.38) ALDH1A1MAPK1TAAR1PYCR1LMNA
SCHEMBL23943395 0.73 ALDH1A1 (0.41) ALDH1A1MAPK1TAAR1GABRA1GABRG2
SCHEMBL10427661 0.73 OPRM1 (0.36) ALDH1A1TAAR1LMNA
SCHEMBL18773999 0.73 TP53 (0.37)
SCHEMBL20048776 0.72 ALDH1A1 (0.39) ALDH1A1MAPK1TAAR1KDM1AC1S
SCHEMBL8281840 0.72 ALDH1A1 (0.40) ALDH1A1MAPK1TAAR1GABRA1GABRG2
SCHEMBL23513694 0.72 CA12 (0.46) ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017136870-A9 HALOALLYLAMINE INDOLE AND AZAINDOLE DERIVATIVE INHIBITORS OF LYSYL OXIDASES AND USES THEREOF PHARMAXIS LTD. (AU) 2018-02-15 WO disclosed
WO-2017136870-A1 HALOALLYLAMINE INDOLE AND AZAINDOLE DERIVATIVE INHIBITORS OF LYSYL OXIDASES AND USES THEREOF PHARMAXIS LTD. (AU) 2017-08-17 WO disclosed