SCHEMBL19255154

SCHEMBL19255154

CCOC(=O)C(C(C)=O)c1cc(C)ccc1[N+](=O)[O-]

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.48
ALDH1A1 P00352 7/20 0.46
TSHR P16473 2/20 0.45
CYP3A4 P08684 1/20 0.45
KMT2A Q03164 2/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
TDP1 Q9NUW8 3/20 0.41
MAPK1 P28482 2/20 0.41
LMNA P02545 3/20 0.40
POLB P06746 2/20 0.40
HPGD P15428 2/20 0.40
GALR2 O43603 1/20 0.40
MITF O75030 1/20 0.40
HSP90AA1 P07900 1/20 0.40
XBP1 P17861 1/20 0.40
CCR6 P51684 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
KDM4E B2RXH2 2/20 0.40
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2566726 0.93 ALDH1A1 (0.52) MAPTALDH1A1TSHRCYP3A4KMT2A
SCHEMBL27340179 0.89 MAPT (0.48) MAPTALDH1A1TSHRCYP3A4KMT2A
SCHEMBL29594753 0.86 KMT2A (0.56) MAPTALDH1A1KMT2ASMN1; SMN2MAPK1
SCHEMBL19211694 0.86 KMT2A (0.56) MAPTALDH1A1KMT2ASMN1; SMN2MAPK1
SCHEMBL19249950 0.85 ALDH3A1 (0.43) MAPTALDH1A1KMT2ASMN1; SMN2TDP1
SCHEMBL7749609 0.81 ALDH1A1 (0.40) MAPTALDH1A1KMT2ASMN1; SMN2TDP1
SCHEMBL492620 0.80 MAPT (0.54) MAPTALDH1A1TSHRKMT2ASMN1; SMN2
SCHEMBL25450873 0.80 ALDH1A1 (0.50) MAPTALDH1A1KMT2ASMN1; SMN2TDP1
SCHEMBL4715558 0.80 ALDH1A1 (0.50) MAPTALDH1A1TSHRKMT2ASMN1; SMN2
SCHEMBL14334237 0.80 ALDH1A1 (0.50) MAPTALDH1A1KMT2ASMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017136870-A9 HALOALLYLAMINE INDOLE AND AZAINDOLE DERIVATIVE INHIBITORS OF LYSYL OXIDASES AND USES THEREOF PHARMAXIS LTD. (AU) 2018-02-15 WO disclosed
WO-2017136870-A1 HALOALLYLAMINE INDOLE AND AZAINDOLE DERIVATIVE INHIBITORS OF LYSYL OXIDASES AND USES THEREOF PHARMAXIS LTD. (AU) 2017-08-17 WO disclosed