SCHEMBL19258920

SCHEMBL19258920

CC(C)NC(=O)c1cc(Br)nc(-c2ccc(F)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.45
ADORA2A P29274 4/20 0.45
SCN9A Q15858 9/20 0.45
ADORA1 P30542 3/20 0.42
ADORA2B P29275 1/20 0.42
RIPK1 Q13546 1/20 0.42
HDAC4 P56524 1/20 0.41
XDH P47989 2/20 0.40
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18824114 0.87 ALOX15 (0.47) ADORA3ADORA2AADORA1ADORA2BRIPK1
SCHEMBL19207313 0.82 NPC1 (0.51) ADORA3ADORA2ASCN9AADORA1NPC1
SCHEMBL18389333 0.82 MAPT (0.46) ADORA3ADORA2ASCN9AADORA1RIPK1
SCHEMBL19207281 0.79 CA12 (0.54) ADORA3ADORA2ASCN9AADORA1ALDH1A1
SCHEMBL19207267 0.79 ADORA3 (0.42) ADORA3ADORA2ASCN9AADORA1NPC1
SCHEMBL19207293 0.78 MAP4K4 (0.48) ADORA3ADORA2ASCN9AADORA1NPC1
SCHEMBL18823914 0.78 ADORA3 (0.44) ADORA3ADORA2ASCN9AADORA1HDAC4
SCHEMBL19259013 0.77 ADORA3 (0.41) ADORA3ADORA2ASCN9AADORA1HDAC4
SCHEMBL19207263 0.77 ADORA3 (0.41) ADORA3ADORA2ASCN9AADORA1HDAC4
SCHEMBL19207307 0.76 HPGDS (0.42) ADORA3ADORA2ASCN9AADORA1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017133990-A1 PYRAZOL-PYRIDINE DERIVATIVES AS EAAT3 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2017-08-10 WO disclosed