SCHEMBL19262174

SCHEMBL19262174

CC(C)[C@H]1C[C@](C#N)(c2cc(F)cc(F)c2)C1

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.33
PDE4B Q07343 2/20 0.33
PDE4C Q08493 2/20 0.33
PDE4D Q08499 2/20 0.33
CCR2 P41597 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19262059 0.84 CCR2 (0.44) PDE4APDE4BPDE4CPDE4DCCR2
SCHEMBL19262093 0.83 CCR2 (0.39) PDE4APDE4BPDE4CPDE4DCCR2
SCHEMBL16591237 0.81 SLC6A3 (0.33) PDE4APDE4BPDE4CPDE4DCCR2
SCHEMBL6994236 0.78 OPRL1 (0.39)
SCHEMBL17985231 0.77 EPAS1 (0.33) PDE4APDE4BPDE4CPDE4D
SCHEMBL16591186 0.77 EPAS1 (0.33) PDE4APDE4BPDE4CPDE4D
SCHEMBL1839257 0.74 OPRM1 (0.34)
SCHEMBL7985502 0.73 SLC6A2 (0.33)
SCHEMBL10270571 0.72 PDE4A (0.35) PDE4APDE4BPDE4CPDE4D
SCHEMBL18742483 0.71 NPC1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9738642-B2 Triazolopyridine ether derivatives and their use in neurological and pyschiatric disorders BRISTOL-MYERS SQUIBB COMPANY (US) 2017-08-22 US disclosed