SCHEMBL1927397

SCHEMBL1927397

CC(C)[C@@H](C(=O)ONS(=O)(=O)c1cccc(C(=O)OC(C)(C)C)c1S(C)(=O)=O)N1C(=O)c2ccccc2C1=O

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.38
KMT2A Q03164 2/20 0.37
PLAU P00749 1/20 0.35
ELANE P08246 1/20 0.35
ALDH1A1 P00352 6/20 0.35
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.33
USP2 O75604 1/20 0.33
HTT P42858 2/20 0.33
BRD4 O60885 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1925203 0.82 TP53 (0.46) TP53KMT2APLAUELANEALDH1A1
SCHEMBL20664182 0.77 KMT2A (0.47) TP53KMT2APLAUELANEALDH1A1
SCHEMBL1925513 0.77 KMT2A (0.47) TP53KMT2APLAUELANEALDH1A1
SCHEMBL1951667 0.77 MMP13 (0.33)
SCHEMBL1951093 0.77 MMP13 (0.33)
SCHEMBL1926037 0.75 KDM4E (0.41) KMT2AELANEALDH1A1HPGDHSD17B10
SCHEMBL1926284 0.74 ALOX15 (0.33) KMT2AMEN1ALOX15
SCHEMBL542373 0.74 TP53 (0.55) TP53KMT2APLAUELANEALDH1A1
SCHEMBL1925201 0.73 PTGS2 (0.43)
SCHEMBL1925775 0.72 TP53 (0.49) TP53KMT2APLAUELANEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2509941-A2 N-ACYLATED HYDROXYLAMINE DERIVATIVES AND O-ACYLATED HYDROXYLAMINE DERIVATIVES The Johns Hopkins University (US) 2012-10-17 EP disclosed
WO-2011071951-A2 N-ACYLOXYSULFONAMIDE AND N-HYDROXY-N-ACYLSULFONAMIDE DERIVATIVES JOHNS HOPKINS UNIVERSITY (US) 2011-06-16 WO disclosed