SCHEMBL19284151

SCHEMBL19284151

Cc1ccc(-c2ccc(C(N3C(=O)C=CC3=O)N3C(=O)C=CC3=O)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 4/20 0.44
GRIA4 P48058 1/20 0.36
FFAR1 O14842 1/20 0.35
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
F2 P00734 1/20 0.33
ELANE P08246 1/20 0.33
CTSG P08311 1/20 0.33
CMA1 P23946 1/20 0.33
CTRC Q99895 1/20 0.33
GAA P10253 1/20 0.33
FAAH O00519 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
CHRNA7 P36544 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL384411 0.73 MGLL (0.44) MGLLCYP2D6HPGDFAAHPKM
SCHEMBL9176987 0.69 MGLL (0.87) MGLLHPGDF2ELANECTSG
SCHEMBL22862085 0.65 MGLL (0.77) MGLLHPGDMEN1KMT2AF2
SCHEMBL197731 0.65 ACHE (0.73) CYP2D6CYP2C9HPGDALOX15CYP2C19
SCHEMBL3287696 0.65 ACHE (0.73) CYP2D6CYP2C9HPGDALOX15CYP2C19
SCHEMBL18661495 0.65 ACHE (0.73) CYP2D6CYP2C9HPGDALOX15CYP2C19
SCHEMBL1132573 0.65 KIF11 (0.45) GRIA4HPGDGAACHRNA7ENPP3
SCHEMBL4394149 0.64 ACHE (0.50) CYP2D6CYP2C9HPGDALOX15CYP2C19
SCHEMBL11978843 0.63 CHRNA7 (0.42) GRIA4FFAR1HRH3CHRNA7ENPP3
SCHEMBL13092431 0.63 CHRNA7 (0.42) GRIA4FFAR1CYP2D6CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230391851-A1 ANTIBODIES THE BINDING SITE GROUP LIMITED (GB) 2023-12-07 US disclosed
EP-3420362-B1 ANTIBODIES THE BINDING SITE GROUP LTD (GB) 2023-03-22 EP disclosed
US-20230080943-A1 ASSAY FOR PLASMA CELL ASSOCIATED DISEASE THE BINDING SITE GROUP LIMITED (GB) 2023-03-16 US disclosed
EP-4123308-A1 MASS SPECTROMETRY KIT The Binding Site Group Limited (GB) 2023-01-25 EP disclosed
EP-3420361-B1 MASS SPECTROMETRY KIT THE BINDING SITE GROUP LTD (GB) 2023-01-04 EP disclosed
EP-3631452-B1 ASSAY FOR PLASMA CELL ASSOCIATED DISEASE THE BINDING SITE GROUP LTD (GB) 2022-07-13 EP disclosed
EP-3631452-A1 ASSAY FOR PLASMA CELL ASSOCIATED DISEASE The Binding Site Group Limited (GB) 2020-04-08 EP disclosed
US-20200096520-A1 ASSAY FOR PLASMA CELL ASSOCIATED DISEASE BINDING SITE GROUP LIMITED, THE (GB) 2020-03-26 US disclosed
US-20190094239-A1 MASS SPECTROMETRY KIT MAYO FOUNDATION FOR MEDICAL EDUCATION AND RESEARCH 2019-03-28 US disclosed
EP-3420362-A1 ANTIBODIES The Binding Site Group Limited (GB) 2019-01-02 EP disclosed
EP-3420361-A1 MASS SPECTROMETRY KIT The Binding Site Group Limited (GB) 2019-01-02 EP disclosed
WO-2018215768-A1 ASSAY FOR PLASMA CELL ASSOCIATED DISEASE THE BINDING SITE GROUP LIMITED (GB) 2018-11-29 WO disclosed
WO-2017144900-A1 MASS SPECTROMETRY KIT THE BINDING SITE GROUP LIMITED (GB) 2017-08-31 WO disclosed
WO-2017144903-A1 ANTIBODIES THE BINDING SITE GROUP LIMITED (GB) 2017-08-31 WO disclosed