SCHEMBL19289878

SCHEMBL19289878

COc1ccc(CN[C@@H](C)I)cc1

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CASR P41180 1/20 0.55
IDO1 P14902 2/20 0.52
AGXT P21549 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
ALDH1A1 P00352 2/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
PKM P14618 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
LMNA P02545 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CHRM2 P08172 1/20 0.49
SLC6A4 P31645 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL278630 0.84 CASR (0.58) CASRIDO1AGXTL3MBTL1ALDH1A1
Hydrochloric Acid SCHEMBL14343449 0.82 CASR (0.57) CASRIDO1AGXTL3MBTL1ALDH1A1
SCHEMBL23995592 0.81 CASR (0.55) CASRIDO1AGXTL3MBTL1ALDH1A1
SCHEMBL8610978 0.81 ALDH1A1 (0.57) CASRL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL19865693 0.79 L3MBTL1 (0.57) CASRL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL22342333 0.79 CASR (0.71) CASRL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL12603587 0.79 CASR (0.71) CASRL3MBTL1ALDH1A1MEN1KMT2A
SCHEMBL30865858 0.79 CASR (0.54) CASRIDO1AGXTL3MBTL1ALDH1A1
SCHEMBL9781346 0.78 CASR (0.53) CASRIDO1AGXTL3MBTL1ALDH1A1
SCHEMBL20502219 0.78 L3MBTL1 (0.56) CASRIDO1AGXTL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2861581-B9 1,2,3,4-Tetrahydroisoquinoline-pyrrolidine derivatives as antagonists of apoptosis (IAPs) for the treatment of cancer. BRISTOL MYERS SQUIBB CO (US) 2017-08-30 EP disclosed