SCHEMBL19304366

SCHEMBL19304366

O=C(/C=C/C1=CNCC=C1)Nc1cn(Cc2cc(F)c(F)c(F)c2)cn1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
EGFR P00533 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20330457 0.74 EGFR (0.42) ALDH1A1MAPTHPGDEGFR
SCHEMBL20169984 0.73 HDAC1 (0.36) ALDH1A1MAPTHPGDEGFR
SCHEMBL21533354 0.72 RIPK1 (0.44) CDK5CDK5R1
SCHEMBL20162136 0.70 HDAC1 (0.41) ALDH1A1MAPTHPGDEGFR
SCHEMBL19304065 0.69 HDAC3 (0.45) ALDH1A1HPGD
SCHEMBL20169940 0.66 HDAC1 (0.51) ALDH1A1MAPTHPGD
SCHEMBL20162176 0.65 TAS2R8 (0.40)
SCHEMBL20331324 0.65 CDK5 (0.35) CDK5CDK5R1
SCHEMBL21518096 0.65 TAS2R8 (0.43) CDK5CDK5R1
SCHEMBL18940396 0.64 JUN (0.40) CDK5CDK5R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017146128-A1 IMIDAZOLYLAMIDE DERIVATIVE 大日本住友製薬株式会社 2017-08-31 WO disclosed