SCHEMBL19347347

SCHEMBL19347347

Cn1c(C(=O)NCCCNC(=O)OC(C)(C)C)cc2c(Cl)c(Cl)ccc21

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.46
PHGDH O43175 10/20 0.46
STK17B O94768 1/20 0.42
STK17A Q9UEE5 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
CNR2 P34972 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19342030 0.96 PHGDH (0.47) DRD2PHGDHKDM4EALDH1A1HSD17B10
SCHEMBL26326346 0.84 PHGDH (0.51) PHGDHKDM4EALDH1A1HSD17B10HPGD
SCHEMBL19343635 0.81 PHGDH (0.55) PHGDHKDM4EALDH1A1HSD17B10HPGD
SCHEMBL19344109 0.79 PHGDH (0.53) PHGDHKDM4EALDH1A1HSD17B10HPGD
SCHEMBL25538844 0.79 PHGDH (0.57) PHGDHHSD17B10
SCHEMBL20793451 0.79 PHGDH (0.53) PHGDHKDM4EALDH1A1HSD17B10HPGD
SCHEMBL19347589 0.78 PHGDH (0.45) PHGDHKDM4EALDH1A1HSD17B10HPGD
SCHEMBL20768544 0.77 PHGDH (0.64) PHGDH
SCHEMBL25535260 0.76 PHGDH (0.44) PHGDHKDM4EALDH1A1HSD17B10HPGD
SCHEMBL25536534 0.76 PHGDH (0.49) PHGDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017156179-A1 3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF RAZE THERAPEUTICS, INC. (US) 2017-09-14 WO disclosed