SCHEMBL19360617

SCHEMBL19360617

CCn1c(C(=O)c2ccc(C(F)(F)F)cc2)cc2cc(C(=O)O)ccc21

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.49
CCR2 P41597 1/20 0.45
GPR35 Q9HC97 1/20 0.43
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41
ACSS2 Q9NR19 1/20 0.41
PPARG P37231 1/20 0.41
EPHX2 P34913 1/20 0.41
TEAD1 P28347 1/20 0.41
TEAD4 Q15561 1/20 0.41
TEAD2 Q15562 1/20 0.41
TEAD3 Q99594 1/20 0.41
CYP2C8 P10632 1/20 0.40
IGFBP3 P17936 1/20 0.40
RORC P51449 2/20 0.40
PTPN1 P18031 1/20 0.39
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
SLC6A2 P23975 1/20 0.38
P2RY14 Q15391 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19360616 0.87 KDM4E (0.48) CCR2ALDH1A1ACSS2PPARGRORC
SCHEMBL18440690 0.86 RORC (0.45) SRD5A2CCR2GPR35ALDH1A1KMT2A
SCHEMBL18440701 0.81 RORC (0.55) SRD5A2CCR2ALDH1A1KMT2AACSS2
SCHEMBL19360395 0.77 RORC (0.65) RORC
SCHEMBL19360584 0.77 RORC (0.48) PPARGEPHX2RORC
SCHEMBL19360594 0.75 RORC (0.42) CCR2ALDH1A1KMT2AACSS2PPARG
SCHEMBL17008986 0.75 PPARG (0.51) PPARGRORC
SCHEMBL20465196 0.75 RORC (0.71) RORC
SCHEMBL20465191 0.74 KMT2A (0.46) GPR35ALDH1A1KMT2AACSS2KDM4E
SCHEMBL18440902 0.74 RAB9A (0.43) ALDH1A1KMT2APPARGRORCKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107531679-B Aromatic amide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-07-02 CN disclosed
CN-107531679-A Aromatic amides analog derivative, its preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2018-01-02 CN disclosed
WO-2017157332-A1 AROMATIC AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATIONS THEREOF 江苏恒瑞医药股份有限公司 2017-09-21 WO disclosed