SCHEMBL19360641

SCHEMBL19360641

CCSc1ccc(CNC(=O)c2ccc3c(c2)cc(CN2CCOCC2)n3CC)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
TSHR P16473 1/20 0.48
LMNA P02545 3/20 0.47
MAPT P10636 3/20 0.46
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
KMT2A Q03164 4/20 0.44
TP53 P04637 2/20 0.43
MLLT1 Q03111 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MAPK1 P28482 2/20 0.42
HDAC4 P56524 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
GALR3 O60755 1/20 0.42
MEN1 O00255 2/20 0.41
ENPP2 Q13822 1/20 0.41
HTT P42858 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
FGB P02675 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19360649 0.91 RORC (0.43) LMNAMAPTKMT2ATP53MLLT1
SCHEMBL19360651 0.90 KMT2A (0.43) MAPTKMT2AHDAC6ENPP2
SCHEMBL19360569 0.86 RORC (0.57)
SCHEMBL19360519 0.78 RORC (0.49) LMNAMAPTTP53MLLT1POLB
SCHEMBL19360531 0.78 RORC (0.58) MAPTPPARG
SCHEMBL19360568 0.77 RORC (0.61)
SCHEMBL22512561 0.76 RORC (0.52)
SCHEMBL19360566 0.76 RORC (0.58)
SCHEMBL19360598 0.76 EPHX2 (0.48) ALDH1A1SMN1; SMN2PPARG
SCHEMBL19360650 0.75 KMT2A (0.42) MAPTKMT2AENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017157332-A1 AROMATIC AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATIONS THEREOF 江苏恒瑞医药股份有限公司 2017-09-21 WO disclosed