SCHEMBL19360645

SCHEMBL19360645

CCSc1ccc(CNC(=O)c2ccc3c(c2)nc(Cc2ccc(OC(F)(F)F)cc2)n3C(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 8/20 0.54
ALDH1A1 P00352 5/20 0.49
HPGD P15428 5/20 0.49
CYP2C9 P11712 3/20 0.49
CYP2C19 P33261 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CNR2 P34972 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
KDM4E B2RXH2 4/20 0.49
GAA P10253 1/20 0.48
CYP3A4 P08684 1/20 0.47
BCHE P06276 1/20 0.45
EPHX2 P34913 3/20 0.45
NR1H4 Q96RI1 1/20 0.45
PPARG P37231 2/20 0.45
PPARA Q07869 2/20 0.45
IDH1 O75874 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19360644 0.88 RORC (0.54) RORCSMN1; SMN2
SCHEMBL28581339 0.87 RORC (0.68) RORC
SCHEMBL19360338 0.85 RORC (0.57) RORC
SCHEMBL19360572 0.82 RORC (0.48) RORCSMN1; SMN2
SCHEMBL19360598 0.79 EPHX2 (0.48) RORCALDH1A1HPGDCYP2C9CYP2C19
SCHEMBL30370139 0.76 RORC (0.83) RORC
SCHEMBL29016570 0.76 RORC (0.83) RORC
SCHEMBL19360477 0.75 RORC (0.69) RORC
SCHEMBL19360481 0.74 RORC (0.67) RORC
SCHEMBL19200968 0.73 RORC (0.54) RORCALDH1A1HPGDCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017157332-A1 AROMATIC AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATIONS THEREOF 江苏恒瑞医药股份有限公司 2017-09-21 WO disclosed