SCHEMBL19366459

SCHEMBL19366459

C1CC(CNC2CC2)CCN1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 10/20 0.44
MAOB P27338 3/20 0.44
MAOA P21397 2/20 0.44
GNAI3 P08754 3/20 0.41
GNAO1 P09471 3/20 0.41
GNAI1 P63096 3/20 0.41
ALOX15 P16050 2/20 0.40
TSHR P16473 1/20 0.40
KDM1B Q8NB78 1/20 0.39
ANPEP P15144 1/20 0.39
ERAP2 Q6P179 1/20 0.39
KCNH2 Q12809 1/20 0.37
EPHX1 P07099 1/20 0.36
EPHX2 P34913 1/20 0.36
PRMT5 O14744 1/20 0.36
WDR77 Q9BQA1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5868698 0.95 KDM1A (0.44) KDM1AMAOBMAOAGNAI3GNAO1
SCHEMBL1009313 0.90 GNAI3 (0.44) KDM1AMAOBMAOAGNAI3GNAO1
SCHEMBL13838034 0.89 RAD52 (0.47) KDM1AMAOBMAOAGNAI3GNAO1
Hydrochloric Acid SCHEMBL4796821 0.88 GNAI3 (0.47) KDM1AMAOBMAOAGNAI3GNAO1
SCHEMBL27911707 0.87 KDM1A (0.44) KDM1AMAOBMAOAGNAI3GNAO1
SCHEMBL4264468 0.86 KDM1A (0.47) KDM1AMAOBMAOAGNAI3GNAO1
SCHEMBL4258478 0.86 KDM1A (0.47) KDM1AMAOBMAOAGNAI3GNAO1
SCHEMBL3307772 0.86 GNAI3 (0.41) KDM1AMAOBMAOAGNAI3GNAO1
SCHEMBL4261850 0.86 KDM1A (0.47) KDM1AMAOBMAOAGNAI3GNAO1
SCHEMBL27804953 0.86 GNAI3 (0.41) KDM1AMAOBMAOAGNAI3GNAO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103857393-A Cyclopropylamines as LSD1 inhibitors GLAXOSMITHKLINE LLC 2014-06-11 CN claimed
US-12281116-B2 HTT modulators for treating Huntington's disease CHDI FOUNDATION, INC. (US) 2025-04-22 US disclosed
EP-4433471-A1 N-(2H-INDAZOL-5-YL)PYRAZINE-2-CARBOXAMIDE DERIVATIVES AND SIMILAR COMPOUNDS AS HTT MODULATORS FOR THE TREATMENT OF HUNTINGTON'S DISEASE CHDI Foundation, Inc. (US) 2024-09-25 EP disclosed
CN-118510769-A HTT modulators for the treatment of huntington's disease CHDI基金会股份有限公司 2024-08-16 CN disclosed
US-20230159531-A1 HTT MODULATORS FOR TREATING HUNTINGTON'S DISEASE CHDI FOUNDATION, INC. 2023-05-25 US disclosed
US-20230159531-A1 HTT MODULATORS FOR TREATING HUNTINGTON'S DISEASE CHDI FOUNDATION, INC. 2023-05-25 US disclosed
US-20230159531-A1 HTT MODULATORS FOR TREATING HUNTINGTON'S DISEASE CHDI FOUNDATION, INC. 2023-05-25 US disclosed
WO-2023091456-A1 N-(2H-INDAZOL-5-YL)PYRAZINE-2-CARBOXAMIDE DERIVATIVES AND SIMILAR COMPOUNDS AS HTT MODULATORS FOR THE TREATMENT OF HUNTINGTON'S DISEASE CHDI FOUNDATION, INC. (US) 2023-05-25 WO disclosed
WO-2023091456-A1 N-(2H-INDAZOL-5-YL)PYRAZINE-2-CARBOXAMIDE DERIVATIVES AND SIMILAR COMPOUNDS AS HTT MODULATORS FOR THE TREATMENT OF HUNTINGTON'S DISEASE CHDI FOUNDATION, INC. (US) 2023-05-25 WO disclosed
EP-3736265-A1 (HETERO)ARYL CYCLOPROPYLAMINE COMPOUNDS AS LSD1 INHIBITORS Oryzon Genomics, S.A. (ES) 2020-11-11 EP disclosed
EP-2768805-B1 (HETERO)ARYL CYCLOPROPYLAMINE COMPOUNDS AS LSD1 INHIBITORS ORYZON GENOMICS SA (ES) 2020-03-25 EP disclosed
EP-2688568-B1 CYCLOPROPYLAMINES AS LSD1 INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2019-06-19 EP disclosed
WO-2017158136-A1 METHODS TO DETERMINE KDM1A TARGET ENGAGEMENT AND CHEMOPROBES USEFUL THEREFOR ORYZON GENOMICS, S.A. (ES) 2017-09-21 WO disclosed
CN-107001318-A N- (hetero) aryl-substituted heterocyclic derivatives useful for the treatment of diseases or disorders associated with the central nervous system 克罗诺斯治疗有限公司 2017-08-01 CN disclosed
CN-103857393-A Cyclopropylamines as LSD1 inhibitors GLAXOSMITHKLINE LLC 2014-06-11 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12281116-B2 HTT modulators for treating Huntington's disease HTT, HYPK, ATXN2 KDM1A 3172/4885MAOB 1600/4885MAOA 1737/4885
US-20230159531-A1 HTT MODULATORS FOR TREATING HUNTINGTON'S DISEASE HTT, HYPK, ATXN2 KDM1A 3172/4885MAOB 1600/4885MAOA 1737/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.