SCHEMBL19370960

SCHEMBL19370960

COc1ccc(CCN2CCC(=O)NC2=O)cc1

nearest known ligand 0.74

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.74
MEN1 O00255 2/20 0.55
ALDH1A1 P00352 2/20 0.55
KMT2A Q03164 2/20 0.55
TSHR P16473 1/20 0.55
SIGMAR1 Q99720 2/20 0.54
HRH3 Q9Y5N1 1/20 0.51
GSK3A P49840 2/20 0.50
GSK3B P49841 2/20 0.50
DAO P14920 1/20 0.50
MAPT P10636 1/20 0.48
DDB1 Q16531 1/20 0.47
CRBN Q96SW2 1/20 0.47
KCNJ1 P48048 1/20 0.46
KCNH2 Q12809 1/20 0.46
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
KCNA5 P22460 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29607421 0.85 GAA (1.00) GAAMEN1ALDH1A1KMT2ASIGMAR1
SCHEMBL11432099 0.82 SIGMAR1 (0.60) GAAMEN1KMT2ASIGMAR1HRH3
SCHEMBL22623804 0.80 DDB1 (0.71) GAAMEN1ALDH1A1KMT2ATSHR
SCHEMBL16429902 0.77 KMT2A (0.64) MEN1ALDH1A1KMT2ASIGMAR1HRH3
SCHEMBL19359333 0.76 POLB (0.59) GAAMEN1ALDH1A1KMT2ATSHR
SCHEMBL19359354 0.76 GAA (0.56) GAAALDH1A1
SCHEMBL3714297 0.73 SIGMAR1 (0.75) MEN1KMT2ASIGMAR1HRH3GSK3A
SCHEMBL28967239 0.73 GSK3A (0.64) GAAMEN1ALDH1A1KMT2ATSHR
SCHEMBL6101068 0.73 GAA (0.73) GAAMEN1ALDH1A1KMT2ASIGMAR1
SCHEMBL19359486 0.72 DDB1 (0.67) GAASIGMAR1GSK3AGSK3BDDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017161119-A1 SMALL MOLECULES AGAINST CEREBLON TO ENHANCE EFFECTOR T CELL FUNCTION H. LEE MOFFITT CANCER CENTER & RESEARCH INSTITUTE, INC. (US) 2017-09-21 WO disclosed