SCHEMBL11432099

SCHEMBL11432099

COc1ccc(CCN2CCC2=O)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.60
HRH3 Q9Y5N1 2/20 0.57
KMT2A Q03164 4/20 0.56
MEN1 O00255 2/20 0.56
TDP1 Q9NUW8 1/20 0.56
GSK3A P49840 2/20 0.55
GSK3B P49841 2/20 0.55
GAA P10253 1/20 0.52
DAO P14920 1/20 0.51
KCNJ1 P48048 1/20 0.50
KCNH2 Q12809 1/20 0.50
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
NPC1 O15118 1/20 0.49
RECQL P46063 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16429902 0.91 KMT2A (0.64) SIGMAR1HRH3KMT2AMEN1TDP1
SCHEMBL11432095 0.83 GAA (0.68) SIGMAR1KMT2AMEN1GSK3AGSK3B
SCHEMBL19370960 0.82 GAA (0.74) SIGMAR1HRH3KMT2AMEN1GSK3A
SCHEMBL11513541 0.78 NPC1 (0.58) SIGMAR1KMT2AMEN1TDP1GSK3A
SCHEMBL28967239 0.77 GSK3A (0.64) SIGMAR1HRH3KMT2AMEN1GSK3A
SCHEMBL3714297 0.77 SIGMAR1 (0.75) SIGMAR1HRH3KMT2AMEN1TDP1
SCHEMBL9491484 0.77 MTNR1A (0.63) HRH3KMT2AMEN1TDP1MAOA
SCHEMBL10195154 0.74 GSK3A (0.64) SIGMAR1HRH3KMT2AMEN1GSK3A
SCHEMBL3459387 0.74 L3MBTL1 (0.64) SIGMAR1HRH3KMT2AMEN1GSK3A
SCHEMBL4509396 0.74 ACACB (0.64) SIGMAR1HRH3KMT2AMEN1GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0023097-A1 De-arylmethylation of N-mono- or N-diarylmethyl-beta-lactams; novel azetizinones having anti-bacterial activity SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1981-01-28 EP disclosed
US-4163743-A Beta-lactams, their production from azetidine carboxylic acids, intermediates thereto and derivatives thereof RESEARCH CORPORATION (US) 1979-08-07 US disclosed