SCHEMBL19404754

SCHEMBL19404754

COc1cc(Br)c(Cl)cc1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 4/20 0.44
POLB P06746 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
PRKDC P78527 1/20 0.39
LCK P06239 1/20 0.38
FYN P06241 1/20 0.38
ALDH1A1 P00352 1/20 0.38
PRNP P04156 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
GAA P10253 1/20 0.38
NPC1 O15118 1/20 0.38
TAAR1 Q96RJ0 2/20 0.37
AHR P35869 2/20 0.37
ALOX5 P09917 1/20 0.36
PTGS2 P35354 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
TSHR P16473 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16384984 0.91 NQO2 (0.41) NQO2POLBL3MBTL1MAPTNPSR1
SCHEMBL29587335 0.84 PRKDC (0.48) POLBL3MBTL1MAPTNPSR1PRKDC
SCHEMBL21403963 0.83 GAA (0.47) NQO2POLBL3MBTL1MAPTNPSR1
SCHEMBL29885672 0.82 NPC1 (0.56) POLBL3MBTL1MAPTNPSR1PRKDC
SCHEMBL263749 0.82 NPC1 (0.56) POLBL3MBTL1MAPTNPSR1PRKDC
SCHEMBL28788044 0.82 HTR2A (0.47) POLBL3MBTL1MAPTNPSR1TAAR1
SCHEMBL12706044 0.81 GAA (0.43) NQO2L3MBTL1MAPTNPSR1ALDH1A1
SCHEMBL16167828 0.81 L3MBTL1 (0.56) NQO2POLBL3MBTL1MAPTNPSR1
SCHEMBL20836401 0.79 MAPT (0.50) NQO2POLBL3MBTL1MAPTNPSR1
SCHEMBL31483694 0.79 MAPT (0.50) NQO2POLBL3MBTL1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021252818-A1 CYCLOPROPYL DIHYDROQUINOLINE SULFONAMIDE COMPOUNDS AMGEN INC. (US) 2021-12-16 WO disclosed
WO-2021252820-A1 CYCLOBUTYL DIHYDROQUINOLINE SULFONAMIDE COMPOUNDS AMGEN INC. (US) 2021-12-16 WO disclosed
WO-2017165139-A1 1,4,5-SUBSTITUTED 1,2,3-TRIAZOLE ANALOGUES AS ANTAGONISTS OF THE PREGNANE X RECEPTOR ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2017-09-28 WO disclosed