SCHEMBL19418249

SCHEMBL19418249

CC(C)C(=O)N(c1ccc(C#N)cc1)C1CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNK O75909 4/20 0.40
CCNA2 P20248 4/20 0.40
CDK2 P24941 4/20 0.40
CDK12 Q9NYV4 4/20 0.40
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
NSD2 O96028 3/20 0.39
PGR P06401 1/20 0.37
NSD3 Q9BZ95 1/20 0.37
PDK2 Q15119 2/20 0.37
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19418280 0.78 CCNK (0.48) CCNKCCNA2CDK2CDK12MEN1
SCHEMBL1539141 0.76 NPC1 (0.42) CCNKCCNA2CDK2CDK12MEN1
SCHEMBL7873766 0.76 CCNK (0.47) CCNKCCNA2CDK2CDK12MEN1
SCHEMBL27808928 0.74 SLC6A4 (0.50) SLC6A2SLC6A4CYP2D6
SCHEMBL28787509 0.74 MEN1 (0.52) MEN1ALDH1A1MAPTTSHRKMT2A
SCHEMBL3081660 0.73 SLC6A2 (0.49) SLC6A2SLC6A4CYP2D6
SCHEMBL21152972 0.71 GPR119 (0.44) CCNKCCNA2CDK2CDK12MEN1
SCHEMBL12733187 0.69 MAOA (0.40) ALDH1A1TSHRSLC6A2SLC6A4NSD2
SCHEMBL19418071 0.68 MAOA (0.39) ALDH1A1TSHRSLC6A2SLC6A4NSD2
SCHEMBL7153765 0.67 CCNK (0.42) CCNKCCNA2CDK2CDK12MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925757-B1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES NOVARTIS AG (CH) 2017-10-04 EP disclosed