Toltrazuril

Toltrazuril

SCHEMBL19436333

Cc1cc(-n2c(=O)[nH]c(=O)n(C)c2=O)ccc1Oc1ccc(SC(F)(F)F)cc1.NC(=O)NC(N)=O

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 12/20 0.49
NTRK2 Q16620 12/20 0.49
IGF1R P08069 4/20 0.49
FGFR1 P11362 4/20 0.49
NTRK3 Q16288 9/20 0.40
BRAF P15056 4/20 0.35
BCAT2 O15382 2/20 0.33
BCAT1 P54687 2/20 0.33
SLC6A4 P31645 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
KIF11 P52732 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Toltrazuril SCHEMBL29509205 0.92 NTRK1 (0.57) NTRK1NTRK2IGF1RFGFR1NTRK3
Toltrazuril SCHEMBL248912 0.92 NTRK1 (0.57) NTRK1NTRK2IGF1RFGFR1NTRK3
Toltrazuril SCHEMBL21812043 0.92 NTRK1 (0.57) NTRK1NTRK2IGF1RFGFR1NTRK3
SCHEMBL13780159 0.84 NTRK1 (0.48) NTRK1NTRK2IGF1RFGFR1NTRK3
SCHEMBL10975351 0.83 NTRK1 (0.52) NTRK1NTRK2IGF1RFGFR1NTRK3
SCHEMBL20328512 0.81 NTRK1 (0.76) NTRK1NTRK2IGF1RFGFR1NTRK3
SCHEMBL10525684 0.81 NTRK1 (0.58) NTRK1NTRK2IGF1RFGFR1NTRK3
SCHEMBL11478539 0.81 NTRK1 (0.45) NTRK1NTRK2IGF1RFGFR1NTRK3
SCHEMBL15783169 0.81 NTRK1 (0.55) NTRK1NTRK2IGF1RFGFR1NTRK3
SCHEMBL10525747 0.79 NTRK1 (0.51) NTRK1NTRK2IGF1RFGFR1NTRK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9802906-B1 Process for the preparation of toltrazuril and an intermediate useful for its preparation ERREGIERRE S.P.A. (IT) 2017-10-31 US disclosed
US-20170291880-A1 PROCESS FOR THE PREPARATION OF TOLTRAZURIL AND AN INTERMEDIATE USEFUL FOR ITS PREPARATION ERREGIERRE S.P.A. (IT) 2017-10-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170291880-A1 PROCESS FOR THE PREPARATION OF TOLTRAZURIL AND AN INTERMEDIATE USEFUL FOR ITS PREPARATION TPMT, TTR, TFPI NTRK1 36/4885NTRK2 476/4885IGF1R 1009/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.