SCHEMBL19440243

SCHEMBL19440243

Cc1cc(C(C)(C)c2cccc(OC(F)(F)F)c2)ccc1C(C)C

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CETP P11597 9/20 0.39
KIF11 P52732 1/20 0.39
CCR6 P51684 2/20 0.36
PDE2A O00408 1/20 0.36
KCNH2 Q12809 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
PLA2G1B P04054 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ATG4B Q9Y4P1 1/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
CARM1 Q86X55 1/20 0.34
GRM5 P41594 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19120701 0.86 SLC22A12 (0.38) CETPKIF11CCR6PDE2AKCNH2
SCHEMBL23252277 0.85 CCR6 (0.38) CETPKIF11CCR6PDE2AKCNH2
SCHEMBL12883121 0.80 PDE2A (0.48) CETPPDE2APLA2G1BTDP1ATG4B
SCHEMBL19275146 0.78 KCNK3 (0.41) PLA2G1BTDP1ATG4BCARM1
SCHEMBL102298 0.73 KIF11 (0.49) CETPKIF11CCR6KCNH2HDAC8
SCHEMBL14997534 0.72 CNR1 (0.36) PDE2A
SCHEMBL21361482 0.71 L3MBTL1 (0.45) KIF11ESR1ESR2
SCHEMBL21974679 0.71 PDE2A (0.38) PDE2ACARM1
SCHEMBL24910303 0.71 CETP (0.40) CETPKCNH2TDP1
SCHEMBL4968089 0.71 KIF11 (0.50) CETPKIF11CCR6KCNH2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9782408-B2 Modulators of cystic fibrosis transmembrane conductance regulator VERTEX PHARMACEUTICALS INCORPORATED (US) 2017-10-10 US disclosed