SCHEMBL19446249

SCHEMBL19446249

CCc1cnc(OC)c(S(=O)(=O)N(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.38
MAPT P10636 3/20 0.38
TSHR P16473 2/20 0.38
GLA P06280 1/20 0.37
ALPL P05186 1/20 0.36
GSTO1 P78417 2/20 0.35
RXFP1 Q9HBX9 1/20 0.34
ALDH1A1 P00352 1/20 0.33
PIK3CD O00329 2/20 0.32
NPC1 O15118 1/20 0.32
TNF P01375 1/20 0.32
RAB9A P51151 1/20 0.32
NOD1 Q9Y239 1/20 0.32
KCNH2 Q12809 1/20 0.32
PIK3R1 P27986 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22548597 0.83 PTGS2 (0.46) PTGS2ALPLPIK3CDPIK3R1PIK3CA
SCHEMBL31535985 0.81 PTGS2 (0.40) PTGS2ALPLALDH1A1PIK3CDPIK3R1
SCHEMBL11918252 0.80 TSHR (0.43) PTGS2MAPTTSHRGLAALPL
SCHEMBL9955416 0.78 TSHR (0.40) MAPTTSHRGLAALPLALDH1A1
SCHEMBL10141687 0.76 TSHR (0.37) MAPTTSHRGLAALPLALDH1A1
SCHEMBL14247505 0.75 TSHR (0.36) MAPTTSHRGLARXFP1ALDH1A1
SCHEMBL20234028 0.70 PIK3CD (0.50) PTGS2PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL9954021 0.70 MAPT (0.43) MAPTTSHRALDH1A1NPC1RAB9A
SCHEMBL9954248 0.70 ALPL (0.54) MAPTTSHRGLAALPL
SCHEMBL12524837 0.70 PTGS2 (0.50) PTGS2PIK3CDNPC1RAB9APIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2516417-B1 ISOINDOLINONE INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE VERTEX PHARMA (US) 2017-10-11 EP disclosed