SCHEMBL19466166

SCHEMBL19466166

O=C(O)Cc1ccc(-c2ccc(=O)[nH]c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCC4 O15439 1/20 0.58
LMNA P02545 1/20 0.58
GAA P10253 1/20 0.58
TSHR P16473 1/20 0.58
PTGS1 P23219 1/20 0.58
HTT P42858 1/20 0.58
CA2 P00918 1/20 0.47
CAMK2A Q9UQM7 1/20 0.47
RXRA P19793 6/20 0.46
RXRB P28702 6/20 0.46
RXRG P48443 6/20 0.46
AKR1B1 P15121 1/20 0.45
FFAR1 O14842 2/20 0.45
PTGS2 P35354 1/20 0.43
NR1H4 Q96RI1 2/20 0.43
RORC P51449 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ENPP2 Q13822 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1972884 0.85 CA2 (0.48) ABCC4LMNAGAATSHRPTGS1
SCHEMBL68027 0.80 LMNA (0.86) ABCC4LMNAGAATSHRPTGS1
SCHEMBL18427891 0.80 LMNA (0.86) ABCC4LMNAGAATSHRPTGS1
SCHEMBL31370206 0.76 SLC7A5 (0.54) LMNAPTGS1PTGS2ALDH1A1HSD17B10
SCHEMBL31477842 0.76 HRH3 (0.56) CA2ALDH1A1
SCHEMBL1867386 0.76 BCL2L1 (0.50) TSHRCA2RXRARXRBRXRG
SCHEMBL694974 0.74 MAPT (0.48) GAAALDH1A1HPGDHSD17B10
Felbinac SCHEMBL26084 0.74 LMNA (1.00) ABCC4LMNAGAATSHRPTGS1
SCHEMBL12126599 0.74 LMNA (0.75) ABCC4LMNAGAATSHRPTGS1
SCHEMBL69614 0.73 CA2 (0.79) ABCC4LMNAGAATSHRPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9789100-B2 Compounds as rearranged during transfection (RET) inhibitors GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-10-17 US disclosed