SCHEMBL19475342

SCHEMBL19475342

Nc1ccc(-c2cc(C(=O)O)c3cc(Cl)ccc3n2)nc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.61
ALDH1A1 P00352 1/20 0.61
ALOX5 P09917 1/20 0.61
CYP2C9 P11712 1/20 0.61
HPGD P15428 1/20 0.61
CASP7 P55210 1/20 0.61
HIF1A Q16665 1/20 0.61
HSD17B10 Q99714 1/20 0.61
DHODH Q02127 7/20 0.56
KMT2A Q03164 3/20 0.50
EPRS1 P07814 1/20 0.50
MAPT P10636 1/20 0.49
KDM4E B2RXH2 1/20 0.47
MOK Q9UQ07 1/20 0.47
MEN1 O00255 2/20 0.47
RXFP1 Q9HBX9 1/20 0.47
PLA2G2A P14555 1/20 0.46
EIF4A1 P60842 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19475331 0.83 ALDH1A1 (0.84) PTGESALDH1A1ALOX5CYP2C9HPGD
SCHEMBL19475339 0.83 NPC1 (0.63) ALDH1A1HPGDHSD17B10DHODHKMT2A
SCHEMBL19475309 0.81 MOK (0.72) ALDH1A1HPGDCASP7HSD17B10KMT2A
SCHEMBL19475455 0.80 ALDH1A1 (0.73) PTGESALDH1A1ALOX5CYP2C9HPGD
SCHEMBL23590223 0.79 KDM4E (0.68) PTGESALDH1A1ALOX5CYP2C9HPGD
SCHEMBL19475402 0.78 HAVCR2 (0.55) ALDH1A1KMT2AMAPTKDM4EMOK
SCHEMBL17211764 0.77 ALDH1A1 (0.69) PTGESALDH1A1ALOX5CYP2C9HPGD
SCHEMBL14286200 0.76 HSD17B10 (1.00) PTGESALDH1A1ALOX5CYP2C9HPGD
SCHEMBL5529524 0.76 HSD17B10 (0.94) PTGESALDH1A1ALOX5CYP2C9HPGD
SCHEMBL23590220 0.76 DHODH (0.67) PTGESALDH1A1ALOX5CYP2C9HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11192859-B2 Quinoline compounds as modulators of RAGE activity and uses thereof UNIV NEW YORK (US) 2021-12-07 US disclosed
US-11192859-B2 Quinoline compounds as modulators of RAGE activity and uses thereof UNIV NEW YORK (US) 2021-12-07 US disclosed
US-20190194136-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF UNIV NEW YORK (US) 2019-06-27 US disclosed
US-20190194136-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF UNIV NEW YORK (US) 2019-06-27 US disclosed
WO-2017184547-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF NEW YORK UNIVERSITY (US) 2017-10-26 WO disclosed
WO-2017184547-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF NEW YORK UNIVERSITY (US) 2017-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190194136-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF AGER, HMGB1, GPR119 PTGES 1213/4885ALDH1A1 1885/4885ALOX5 1110/4885
US-11192859-B2 Quinoline compounds as modulators of RAGE activity and uses thereof AGER, HMGB1, GPR119 PTGES 1213/4885ALDH1A1 1885/4885ALOX5 1110/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.