Brucine

Brucine

SCHEMBL19476145

COc1cc2c(cc1OC)C13CCN4CC5=CCO[C@H]6CC(=O)N2[C@H]1[C@H]6[C@H]5CC43

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAS2R10 Q9NYW0 2/20 1.00
CHRM1 P11229 1/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
GLRA1 P23415 14/20 0.73
GLRB P48167 14/20 0.73
CYP3A4 P08684 2/20 0.71
MEN1 O00255 2/20 0.71
KMT2A Q03164 2/20 0.71
SCN1A P35498 1/20 0.71
TAS2R46 P59540 1/20 0.71
SCN2A Q99250 1/20 0.71
SCN3A Q9NY46 1/20 0.71
CYP1A2 P05177 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Brucine SCHEMBL113229 1.00 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL29391712 1.00 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL1648976 1.00 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL10307298 1.00 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL14029321 1.00 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL23468158 1.00 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL12293782 1.00 TAS2R10 (1.00) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL6233075 0.99 TAS2R10 (0.98) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL6794678 0.99 TAS2R10 (0.98) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB
Brucine SCHEMBL7253414 0.99 TAS2R10 (0.98) TAS2R10CHRM1SMN1; SMN2GLRA1GLRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017180248-A1 ENANTIOENRICHED VIRIDICATUMTOXIN B ANALOGS WILLIAM MARSH RICE UNIVERSITY (US) 2017-10-19 WO disclosed