SCHEMBL19476245

SCHEMBL19476245

COc1cc2c(c(OCc3ccc(C(F)(F)F)cc3)c1)C(=O)c1c(O)ccc(OCc3ccccc3)c1C2

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PSEN1 P49768 6/20 0.42
ALOX5 P09917 4/20 0.42
PPARG P37231 2/20 0.42
PTGES O14684 1/20 0.42
PTPN1 P18031 5/20 0.41
PTPN2 P17706 2/20 0.41
PTPN6 P29350 2/20 0.41
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
SLC2A1 P11166 1/20 0.39
FFAR4 Q5NUL3 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
ACHE P22303 1/20 0.38
KEAP1 Q14145 1/20 0.38
NFE2L2 Q16236 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19476060 0.94 MAOB (0.39) PSEN1ALOX5PTPN1PTPN2PTPN6
SCHEMBL19476244 0.90 PSEN1 (0.46) PSEN1ALOX5PPARGPTGES
SCHEMBL19175928 0.89 CA1 (0.45) PPARGCA1CA2ACHE
SCHEMBL19476035 0.84 CA1 (0.39) MAOBCA1CA2ACHE
SCHEMBL19476241 0.83 CA1 (0.39) PTPN1CA1CA2ACHE
SCHEMBL19168589 0.80 NPC1 (0.40) MAOBFFAR4
SCHEMBL19476057 0.78 MAOB (0.48) PTPN1MAOAMAOB
SCHEMBL19476171 0.74 PARP15 (0.46) CA1CA2KEAP1NFE2L2
SCHEMBL17469676 0.72 CES2 (0.40) CA1CA2ACHE
SCHEMBL19476170 0.72 KDM4E (0.47) ALOX5CA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017180248-A1 ENANTIOENRICHED VIRIDICATUMTOXIN B ANALOGS WILLIAM MARSH RICE UNIVERSITY (US) 2017-10-19 WO disclosed