SCHEMBL19478673

SCHEMBL19478673

CCCCCc1ccc2nc(C)c(C)nc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 2/20 0.52
TLR8 Q9NR97 6/20 0.48
S1PR4 O95977 1/20 0.44
S1PR1 P21453 1/20 0.44
S1PR5 Q9H228 1/20 0.44
SKP2 Q13309 1/20 0.43
ESR1 P03372 2/20 0.43
ADRA2A P08913 2/20 0.43
ADORA3 P0DMS8 2/20 0.43
TACR2 P21452 2/20 0.43
SLC6A2 P23975 2/20 0.43
SLC6A4 P31645 2/20 0.43
SLC6A3 Q01959 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
SHBG P04278 1/20 0.43
TP53 P04637 1/20 0.43
CYP3A4 P08684 1/20 0.43
HSPD1 P10809 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23130637 0.95 PSMB5 (0.57) PSMB5TLR8SKP2LMNATP53
SCHEMBL18805360 0.87 TLR8 (0.51) TLR8S1PR4S1PR1S1PR5ESR1
SCHEMBL13156563 0.87 TLR8 (0.51) TLR8S1PR4S1PR1S1PR5ESR1
SCHEMBL7073871 0.80 PSMB5 (0.54) PSMB5TLR8SKP2KDM4EALDH1A1
SCHEMBL6077149 0.80 PSMB5 (0.48) PSMB5TLR8S1PR4S1PR1S1PR5
SCHEMBL6910786 0.79 TLR8 (0.51) TLR8S1PR4S1PR1S1PR5SKP2
SCHEMBL19992509 0.79 SMN1; SMN2 (0.46) KDM4EALDH1A1LMNATP53CYP3A4
SCHEMBL5154662 0.78 TDP1 (0.42) PSMB5KDM4EALDH1A1CYP3A4HIF1A
SCHEMBL12846225 0.76 TLR8 (0.45) PSMB5TLR8S1PR4S1PR1S1PR5
SCHEMBL6347222 0.75 ESR1 (0.47) TLR8ESR1ADRA2AADORA3TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017178828-A1 CONJUGATES AND CONJUGATING REAGENTS COMPRISING A LINKER THAT INCLUDES AT LEAST TWO (-CH2-CH2-0-) UNITS IN A RING POLYTHERICS LIMITED (GB) 2017-10-19 WO disclosed