SCHEMBL19480883

SCHEMBL19480883

Cn1ccc(-c2cccnc2N)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.46
KMT2A Q03164 1/20 0.44
CASP6 P55212 1/20 0.43
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
NOS2 P35228 1/20 0.42
MAP4K4 O95819 1/20 0.42
ADORA2A P29274 2/20 0.40
MKNK1 Q9BUB5 2/20 0.39
MKNK2 Q9HBH9 2/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
TGFBR1 P36897 1/20 0.39
AKT1 P31749 1/20 0.38
AKT2 P31751 1/20 0.38
SYK P43405 1/20 0.38
NTRK1 P04629 1/20 0.37
LRRK2 Q5S007 1/20 0.37
JMJD6 Q6NYC1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15885475 0.80 CASP6 (0.47) KEAP1KMT2ACASP6MKNK1MKNK2
SCHEMBL22940968 0.79 CASP6 (0.49) KEAP1KMT2ACASP6ADORA2AADRA1D
SCHEMBL1850624 0.79 KMT2A (0.44) KEAP1KMT2ACASP6ADRA1DADRA1A
SCHEMBL22940967 0.76 RAB9A (0.47) KMT2ACASP6JMJD6JAK2JAK3
SCHEMBL22230356 0.76 KEAP1 (0.50) KEAP1KMT2AADORA2ATGFBR1JMJD6
SCHEMBL11377293 0.76 KMT2A (0.53) KEAP1KMT2AADRA1DADRA1AADRA1B
SCHEMBL30211937 0.75 KEAP1 (0.46) KEAP1KMT2ACASP6ADORA2ATGFBR1
SCHEMBL4240350 0.74 MAP4K4 (0.40) NOS3NOS1NOS2MAP4K4MKNK1
SCHEMBL10062975 0.73 MAP4K4 (0.59) KMT2ANOS3NOS1NOS2MAP4K4
SCHEMBL17812984 0.72 KMT2A (0.54) KEAP1KMT2ACASP6NTRK1JMJD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4126844-A1 AMIDE COMPOUNDS AND USES THEREOF Hutchison Medipharma Limited (CN) 2023-02-08 EP disclosed
WO-2021197276-A1 Amide compounds and uses thereof HUTCHISON MEDIPHARMA LIMITED (CN) 2021-10-07 WO disclosed
WO-2017178344-A1 NOVEL N-[(HETEROARYLOXY)PROPANYL]HETEROARYL CARBOXAMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2017-10-19 WO disclosed