SCHEMBL19488778

SCHEMBL19488778

C#Cc1ccc2[nH]c([C@@H]3CCC[C@H](C)N3C(=O)OC(C)(C)C)nc2c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 3/20 0.39
GABRB3 P28472 3/20 0.39
GABRA5 P31644 3/20 0.39
GABRA6 Q16445 3/20 0.39
GABRA4 P48169 2/20 0.39
GABRA1 P14867 2/20 0.39
GABRA2 P47869 2/20 0.39
GABRA3 P34903 1/20 0.39
KAT2B Q92831 1/20 0.33
HCRTR1 O43613 5/20 0.33
HCRTR2 O43614 5/20 0.33
PTGES O14684 2/20 0.33
GPR119 Q8TDV5 1/20 0.33
JAK1 P23458 1/20 0.33
PRCP P42785 1/20 0.32
CHEK2 O96017 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10200239 0.95 GABRG2 (0.40) GABRG2GABRB3GABRA5GABRA6GABRA4
SCHEMBL571669 0.85 PTGES (0.44) GABRG2GABRB3GABRA5GABRA6GABRA4
SCHEMBL571668 0.85 PTGES (0.44) GABRG2GABRB3GABRA5GABRA6GABRA4
SCHEMBL12373570 0.83 GABRA1 (0.42) GABRG2GABRB3GABRA5GABRA6GABRA4
SCHEMBL10201501 0.83 GABRG2 (0.39) GABRG2GABRB3GABRA5GABRA6GABRA4
SCHEMBL12373582 0.83 GABRG2 (0.39) GABRG2GABRB3GABRA5GABRA6GABRA4
SCHEMBL12373508 0.81 HCRTR1 (0.37) HCRTR1HCRTR2JAK1CHEK2
SCHEMBL12373604 0.80 GABRG2 (0.35) GABRG2GABRB3GABRA5GABRA6GABRA4
SCHEMBL12558673 0.79 GABRG2 (0.39) GABRG2GABRB3GABRA5GABRA6GABRA4
SCHEMBL12558668 0.79 HCRTR1 (0.43) HCRTR1HCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2601188-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-10-18 EP disclosed