SCHEMBL19503552

SCHEMBL19503552

C=C1NC(=O)CCC1N1Cc2cc(OC)ccc2C1=C

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
WIZ O95785 1/20 0.45
CRBN Q96SW2 13/20 0.44
IKZF2 Q9UKS7 6/20 0.43
CSNK1A1 P48729 2/20 0.43
METAP1 P53582 1/20 0.42
DDB1 Q16531 3/20 0.41
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19503564 0.88 POLB (0.43) CRBNIKZF2CSNK1A1
SCHEMBL17552859 0.80 CRBN (0.69) WIZCRBNIKZF2CSNK1A1
SCHEMBL24319331 0.80 CRBN (0.69) WIZCRBNIKZF2CSNK1A1
SCHEMBL24891513 0.77 IKZF2 (0.45) CRBNIKZF2
SCHEMBL27117194 0.77 WIZ (0.40) WIZCRBNIKZF2
SCHEMBL25993290 0.76 CRBN (0.55) WIZCRBNIKZF2
SCHEMBL26000355 0.76 CRBN (0.54) WIZCRBNIKZF2
SCHEMBL19503553 0.74 CRBN (0.47) CRBNDDB1
SCHEMBL26022267 0.74 IKZF2 (0.52) WIZCRBNIKZF2
SCHEMBL25994256 0.74 HRH3 (0.36) WIZCRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3820573-B1 3-(5-HYDROXY-1-OXOISOINDOLIN-2-YL)PIPERIDINE-2,6-DIONE DERIVATIVES AND THEIR USE IN THE TREATMENT OF IKAROS FAMILY ZINC FINGER 2 (IKZF2)-DEPENDENT DISEASES NOVARTIS AG (CH) 2023-08-09 EP disclosed
WO-2017184995-A1 COMPOUNDS THAT INDUCE DEGRADATION OF ANTI-APOPTOTIC BCL-2 FAMILY PROTEINS AND THE USES THEREOF BIOVENTURES, LLC (US) 2017-10-26 WO disclosed