SCHEMBL19503752

SCHEMBL19503752

CCCc1nc(C)[nH]c(=O)c1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.46
CDK4 P11802 2/20 0.45
CCND1 P24385 2/20 0.45
ALDH1A1 P00352 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPK1 P28482 1/20 0.38
GLA P06280 1/20 0.35
PARP1 P09874 4/20 0.35
TNKS2 Q9H2K2 1/20 0.35
HPGD P15428 1/20 0.35
USP2 O75604 1/20 0.35
POLB P06746 1/20 0.35
TSHR P16473 1/20 0.35
CCNE2 O96020 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
RAB9A P51151 1/20 0.34
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
BACE1 P56817 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12176674 0.89 HTT (0.43) HTTCDK4CCND1ALDH1A1L3MBTL1
SCHEMBL20990600 0.81 POLB (0.52) HTTCDK4CCND1ALDH1A1L3MBTL1
SCHEMBL9879082 0.78 HTT (0.77) HTTALDH1A1L3MBTL1HPGDUSP2
SCHEMBL19503753 0.78 CDK4 (0.39) HTTCDK4CCND1ALDH1A1L3MBTL1
SCHEMBL5851856 0.74 SMPD3 (0.34) CDK4CCND1ALDH1A1GLAPOLB
SCHEMBL3704415 0.72 PDK2 (0.37) CDK4CCND1ALDH1A1GLAUSP2
SCHEMBL4128983 0.72 PDE2A (0.40) CDK4CCND1ALDH1A1L3MBTL1GLA
SCHEMBL8459493 0.71 KDM4E (0.34) CDK4CCND1ALDH1A1USP2POLB
SCHEMBL3845619 0.70 PDE5A (0.62) ALDH1A1HPGDPOLBPDE3BPDE3A
SCHEMBL172127 0.69 ALDH1A1 (0.58) ALDH1A1L3MBTL1MAPK1GLAPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017184999-A1 EZH2 INHIBITORS AND USES THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2017-10-26 WO disclosed