SCHEMBL19514014

SCHEMBL19514014

CCc1nn2ccc(Cl)cc2c1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FABP4 P15090 2/20 0.42
FABP5 Q01469 2/20 0.42
FABP3 P05413 1/20 0.42
MAT2A P31153 3/20 0.38
LMNA P02545 1/20 0.37
SLC22A12 Q96S37 2/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
KMO O15229 3/20 0.36
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK10 P53779 1/20 0.36
PRMT5 O14744 1/20 0.35
CYP1A2 P05177 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 1/20 0.34
PKM P14618 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19531526 0.84 LMNA (0.46) LMNAMEN1KMT2APKMKDM4E
SCHEMBL28437880 0.83 GABRP (0.38) FABP4FABP5FABP3SLC22A12MEN1
SCHEMBL21584617 0.83 PTGDR2 (0.37) FABP4FABP5FABP3SLC22A12PTGDR2
SCHEMBL19514077 0.79 TP53 (0.44) LMNAKMT2ANPC1RAB9AKDM4E
SCHEMBL2035471 0.78 EGFR (0.48) FABP4FABP5FABP3LMNACYP1A2
SCHEMBL19514080 0.77 NR1H4 (0.46) PTGDR2MEN1KMT2AKDM4E
SCHEMBL19514013 0.76 CYP3A4 (0.47) MEN1KMT2ANPC1RAB9AKDM4E
SCHEMBL21838150 0.74 GABRP (0.38) FABP4FABP5FABP3LMNASLC22A12
SCHEMBL19514081 0.74 ALDH1A1 (0.47) LMNAMEN1KMT2ARAB9A
SCHEMBL19538745 0.74 PTGDR2 (0.48) LMNAPTGDR2CYP1A2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170313697-A1 PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AND USE THEREOF GUANGDONG GOOD MEDICINE AND HEALTH TECHNOLOGY CO., LTD (CN) 2017-11-02 US disclosed
US-20170313697-A1 PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AND USE THEREOF GUANGDONG GOOD MEDICINE AND HEALTH TECHNOLOGY CO., LTD (CN) 2017-11-02 US disclosed
US-20170313697-A1 PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AND USE THEREOF GUANGDONG GOOD MEDICINE AND HEALTH TECHNOLOGY CO., LTD (CN) 2017-11-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170313697-A1 PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AND USE THEREOF ABCG2, ABCC1, PNPO FABP4 4050/4885FABP5 3107/4885FABP3 3408/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.