SCHEMBL1954342

SCHEMBL1954342

CN(C)N1CCC(=O)CC1

nearest known ligand 0.33

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TRIM24 O15164 2/20 0.33
TRIM33 Q9UPN9 2/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trimethylammonium SCHEMBL27932051 0.71
SCHEMBL1577820 0.71
SCHEMBL68353 0.67
SCHEMBL11028940 0.67 MAOA (0.40) TRIM24TRIM33ALDH1A1
SCHEMBL12360481 0.67 BRD4 (0.39) TRIM24TRIM33ALDH1A1
SCHEMBL1955321 0.67 CHRNA7 (0.50)
SCHEMBL1958525 0.67
SCHEMBL4189631 0.65
SCHEMBL2306907 0.65
SCHEMBL378435 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160122342-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2016-05-05 US disclosed
EP-3004096-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2016-04-13 EP disclosed
WO-2014195919-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED (GB) 2014-12-11 WO disclosed
US-8703165-B2 Spiro fused 1-amino-piperdine pyrrolidine dione derivatives with pesticidal activity SYNGENTA CROP PROTECTION, INC. (US) 2014-04-22 US disclosed
EP-2507240-B1 SPIRO FUSED 1-AMINO-PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2014-01-15 EP disclosed
US-8541343-B2 Chemical compounds and their use as pesticides SYNGENTA CROP PROTECTION, INC. (US) 2013-09-24 US disclosed
EP-2507214-A1 CHEMICAL COMPOUNDS AND THEIR USE AS PESTICIDES Syngenta Participations AG (CH) 2012-10-10 EP disclosed
EP-2507240-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY Syngenta Participations AG (CH) 2012-10-10 EP disclosed
US-20120245026-A1 SPIRO FUSED 1-AMINO - PIPERDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA CROP PROTECTION LLC (US) 2012-09-27 US disclosed
US-20120238452-A1 CHEMICAL COMPOUNDS AND THEIR USE AS PESTICIDES SYNGENTA CROP PROTECTION LLC (US) 2012-09-20 US disclosed
WO-2011067135-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067203-A1 CHEMICAL COMPOUNDS AND THEIR USE AS PESTICIDES SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
WO-2011067240-A1 SPIRO FUSED 1 -AMINO - PIPERIDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY SYNGENTA PARTICIPATIONS AG (CH) 2011-06-09 WO disclosed
US-20090233910-A1 Npy antagonists, preparation and uses CEREP (FR) 2009-09-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120245026-A1 SPIRO FUSED 1-AMINO - PIPERDINE PYRROLIDINE DIONE DERIVATIVES WITH PESTICIDAL ACTIVITY DDT, CAT, AQP1 TRIM24 3938/4885TRIM33 4262/4885ALDH1A1 79/4885
US-20120238452-A1 CHEMICAL COMPOUNDS AND THEIR USE AS PESTICIDES DDT, ACHE, CYP1A1 TRIM24 4205/4885TRIM33 3465/4885ALDH1A1 140/4885
US-20090233910-A1 Npy antagonists, preparation and uses NPY1R, NPY5R, NPY2R TRIM24 4038/4885TRIM33 3866/4885ALDH1A1 4542/4885
US-20160122342-A1 ENHANCER OF ZESTE HOMOLOG 2 INHIBITORS EZH2, BMI1, EZH1 TRIM24 1482/4885TRIM33 2521/4885ALDH1A1 2517/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.