SCHEMBL19554282

SCHEMBL19554282

O=C(O)c1ccc2cc(OC(F)(F)Br)ccc2c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.59
PTPN1 P18031 1/20 0.50
ALDH1A1 P00352 2/20 0.45
HSD17B10 Q99714 2/20 0.45
TSHR P16473 1/20 0.45
PIM1 P11309 1/20 0.44
PLA2G2D Q9UNK4 1/20 0.42
RARB P10826 6/20 0.41
RARG P13631 6/20 0.41
RARA P10276 5/20 0.41
MRGPRX4 Q96LA9 2/20 0.41
AURKA O14965 1/20 0.41
TPX2 Q9ULW0 1/20 0.41
CYP26A1 O43174 1/20 0.41
CYP26B1 Q9NR63 1/20 0.41
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
FAAH O00519 1/20 0.40
EPHX2 P34913 1/20 0.40
CYP1A2 P05177 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19554192 0.88 KDM4E (0.61) KDM4EPTPN1ALDH1A1HSD17B10TSHR
SCHEMBL19554294 0.82 NOTUM (0.51) KDM4EALDH1A1MRGPRX4CA1CA2
SCHEMBL19554267 0.79 KDM4E (0.62) KDM4EPTPN1ALDH1A1HSD17B10TSHR
SCHEMBL6916181 0.77 KDM4E (0.68) KDM4EPTPN1ALDH1A1HSD17B10TSHR
SCHEMBL29359975 0.77 KDM4E (0.68) KDM4EPTPN1ALDH1A1HSD17B10TSHR
SCHEMBL29594563 0.77 KDM4E (0.68) KDM4EPTPN1ALDH1A1HSD17B10TSHR
SCHEMBL18758 0.77 KDM4E (0.68) KDM4EPTPN1ALDH1A1HSD17B10TSHR
SCHEMBL8080613 0.76 KDM4E (0.69) KDM4EALDH1A1HPGD
SCHEMBL18288105 0.76 KDM4E (0.58) KDM4EALDH1A1HSD17B10TSHRRARB
Terephthalic Acid SCHEMBL2846917 0.74 TSHR (0.67) KDM4EPTPN1ALDH1A1HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017192304-A1 ARYLCARBOXAMIDES AND USES THEREOF INCEPTION 1, INC. (US) 2017-11-09 WO disclosed