SCHEMBL1958368

SCHEMBL1958368

N[C@@H](CC(=O)O)c1cccs1.O=C(O)C[C@H](NC(=O)OCc1ccccc1)c1cccs1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 10/20 0.44
CTRB1 P17538 2/20 0.42
CASP3 P42574 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2479865 0.93 CASP1 (0.49) CASP1CTRB1CASP3
SCHEMBL2479868 0.93 CASP1 (0.49) CASP1CTRB1CASP3
SCHEMBL27850286 0.81 ATM (0.46) CTRB1
SCHEMBL8417460 0.78 ALDH1A1 (0.49) CTRB1
SCHEMBL2030179 0.78 ALOX5 (0.44)
SCHEMBL2481473 0.78 ALOX5 (0.44)
SCHEMBL3351265 0.78 ALOX5 (0.44)
SCHEMBL11475132 0.76 ATM (0.53) CTRB1HDAC3HDAC1HDAC2
SCHEMBL6955527 0.75 CASP1 (0.60) CASP1CTRB1
SCHEMBL6156731 0.75 CASP1 (0.60) CASP1CTRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011068561-A1 SULFONAMIDE DERIVATIVES AS BCL-2-SELECTIVE APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE DISEASES ABBOTT LABORATORIES (US) 2011-06-09 WO disclosed