SCHEMBL196018

SCHEMBL196018

Nc1nc(=O)[nH]c2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.58
ALDH1A1 P00352 5/20 0.58
HSD17B10 Q99714 3/20 0.58
HPGD P15428 2/20 0.58
TSHR P16473 1/20 0.58
GAA P10253 2/20 0.50
PDPK1 O15530 1/20 0.50
CYP3A4 P08684 1/20 0.50
APP P05067 2/20 0.49
LMNA P02545 2/20 0.48
GLA P06280 1/20 0.48
HTT P42858 1/20 0.48
ATM Q13315 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
ADORA3 P0DMS8 3/20 0.47
PLAUR Q03405 1/20 0.47
CA5A P35218 1/20 0.46
GPR3 P46089 2/20 0.45
PARP1 P09874 2/20 0.45
MEN1 O00255 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29844822 1.00 KDM4E (0.58) KDM4EALDH1A1HSD17B10HPGDTSHR
Pyrazole SCHEMBL28116372 0.86 KDM4E (0.45) KDM4EALDH1A1HSD17B10HPGDTSHR
SCHEMBL2222578 0.77 TYMS (0.50) KDM4EALDH1A1HSD17B10HPGDTSHR
SCHEMBL6099088 0.76 KDM4E (0.58) KDM4EALDH1A1HSD17B10HPGDTSHR
SCHEMBL554709 0.76 KDM4E (0.58) KDM4EALDH1A1HSD17B10HPGDTSHR
SCHEMBL1621540 0.76 GAA (0.50) KDM4EALDH1A1HSD17B10HPGDTSHR
SCHEMBL6076792 0.76 KDM4E (0.58) KDM4EALDH1A1HSD17B10HPGDTSHR
SCHEMBL3139711 0.76 KDM4E (0.58) KDM4EALDH1A1HSD17B10HPGDTSHR
SCHEMBL4413903 0.76 KDM4E (0.58) KDM4EALDH1A1HSD17B10HPGDTSHR
SCHEMBL530191 0.76 ALDH1A1 (0.58) KDM4EALDH1A1HSD17B10HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 567 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12404269-B2 Aminoquinazolinone and aminoisoquinolinone derivatives and application thereof ZHEJIANG UNIVERSITY (CN) 2025-09-02 US claimed
CN-117209437-A Preparation method of aminoquinazolinone derivative 宁夏大学 2023-12-12 CN claimed
CN-109503550-B 2-azaaryl-6-substituted amino quinazolinone compound and preparation method and application thereof 江西师范大学 2022-11-29 CN claimed
US-20220017505-A1 AMINOQUINAZOLINONE AND AMINOISOQUINOLINONE DERIVATIVES AND APPLICATION THEREOF SHANGHAI INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF SCIENCES (CN) 2022-01-20 US claimed
EP-3904343-A1 AMINO QUINAZOLINONE, AMINO ISOQUINOLONE DERIVATIVES AND APPLICATION THEREOF Zhejiang University (CN) 2021-11-03 EP claimed
CN-109516961-B Aminoquinazolinone and aminoisoquinolinone derivatives and uses thereof 浙江大学 2021-01-01 CN claimed
WO-2020134921-A1 AMINO QUINAZOLINONE, AMINO ISOQUINOLONE DERIVATIVES AND APPLICATION THEREOF 浙江大学 2020-07-02 WO claimed
CN-109516961-A Aminoquinazolinone and aminoisoquinoline ketone derivatives and its application 浙江大学 2019-03-26 CN claimed
CN-1302801-B Substituted aminoquinazolinone (thione) derivatives or salts thereof, intermediates thereof, and pest control agents and methods of using the same NIHOU NOHYAKU CO LTD 2013-03-20 CN claimed
US-8034931-B2 Process for producing substituted aminoquinazolinone derivative, intermediate therefor, and pest control agent NIHON NOHYAKU CO., LTD. (JP) 2011-10-11 US claimed
CN-1092188-C Substituted aminoquinazolinone (thione) derivatives or salts thereof, intermediates thereof, and pest control agents and methods of using the same NIHON NOHYAKU CO LTD (JP) 2002-10-09 CN claimed
US-6455535-B1 INSECTICIDES NIHON NOHYAKU CO., LTD. (JP) 2002-09-24 US claimed
EP-0735035-B1 Substituted aminoquinazolinone (thione) derivatives or salts thereof, intermediates thereof, and pest controllers and a method for using the same NIHON NOHYAKU CO LTD (JP) 2002-06-05 EP claimed
CN-1302801-A Substituted aminoquinazolinone (thione) derivatives or salts thereof, intermediates thereof, and pest control agents and methods of using the same NIHOU NOHYAKU CO LTD (JP) 2001-07-11 CN claimed
EP-1097932-A1 Substituted aminoquinazolinone (thione) derivatives or salts thereof, intermediates thereof, and pest controllers and a method for using the same NIHON NOHYAKU CO., LTD. (JP) 2001-05-09 EP claimed
CN-1282517-A Pest controlling agent containing substituted aminoquinazolone or thioketone derivative or its salt as active component NIHON NOHYAKU CO LTD (JP) 2001-02-07 CN claimed
EP-0987255-A2 Substituted aminoquinazolinone (thione) derivatives NIHON NOHYAKU CO., LTD. (JP) 2000-03-22 EP claimed
US-5714492-A INSECTICIDES NIHON NOHYAKU CO., LTD. (JP) 1998-02-03 US claimed
CN-1134933-A Substituted aminoquinazolinone (thione) derivatives or salts thereof, intermediates thereof, and pest control agents and methods of using the same NIHON NOHYAKU CO LTD (JP) 1996-11-06 CN claimed
EP-0735035-A1 Substituted aminoquinazolinone (thione) derivatives or salts thereof, intermediates thereof, and pest controllers and a method for using the same NIHON NOHYAKU CO., LTD. (JP) 1996-10-02 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12404269-B2 Aminoquinazolinone and aminoisoquinolinone derivatives and application thereof PIK3R5, PIK3CA, PIK3R1 KDM4E 1579/4885ALDH1A1 2788/4885HSD17B10 1294/4885
US-20220017505-A1 AMINOQUINAZOLINONE AND AMINOISOQUINOLINONE DERIVATIVES AND APPLICATION THEREOF PIK3R5, PIK3CA, PIK3R1 KDM4E 1579/4885ALDH1A1 2788/4885HSD17B10 1294/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.