SCHEMBL19610482

SCHEMBL19610482

CN1CCC[C@@H](n2ccc(I)n2)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 2/20 0.37
TMEM97 Q5BJF2 1/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SIGMAR1 Q99720 2/20 0.33
KAT2B Q92831 1/20 0.33
ADRA1A P35348 2/20 0.33
HRH1 P35367 2/20 0.33
ADRA1B P35368 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
HTR6 P50406 3/20 0.32
CHRM2 P08172 3/20 0.32
CHRM1 P11229 3/20 0.32
CHRM3 P20309 3/20 0.32
CHRM4 P08173 2/20 0.32
CHRM5 P08912 2/20 0.32
DRD2 P14416 2/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
KCNH2 Q12809 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6221771 1.00 HTR2B (0.37) HTR2BTMEM97ATML3MBTL1SIGMAR1
SCHEMBL15416227 0.83 OPRM1 (0.30) OPRM1
SCHEMBL5800638 0.80 GAA (0.40) L3MBTL1SIGMAR1CHRM2CHRM3HTR2A
SCHEMBL26101147 0.79 SIGMAR1 (0.36) SIGMAR1
SCHEMBL27568268 0.79 SIGMAR1 (0.39) SIGMAR1KCNH2
SCHEMBL28752477 0.78 SIGMAR1 (0.40) SIGMAR1KAT2B
SCHEMBL27586657 0.78 SIGMAR1 (0.40) SIGMAR1KAT2B
SCHEMBL15825704 0.75
SCHEMBL5801362 0.75 HTR3E (0.37) L3MBTL1SIGMAR1IRAK4KCNH2HRH3
SCHEMBL29490572 0.72 GAA (0.36) KAT2BHRH1HTR6CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246327-A1 3-ACETYLENYL-PYRAZOLE-PYRIMIDINE DERIVATIVE, AND PREPARATION METHOD THEREFOR AND USES THEREOF Si Chuan University (CN) 2017-11-22 EP disclosed