SCHEMBL1961273

SCHEMBL1961273

O=C1CCC(N2Cc3cccc(C(=O)NC(=O)Nc4ccc5ccccc5c4)c3C2=O)C(=O)N1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 16/20 0.54
CSNK1A1 P48729 9/20 0.54
IKZF2 Q9UKS7 7/20 0.45
DDB1 Q16531 2/20 0.45
POLB P06746 1/20 0.45
GSPT1 P15170 1/20 0.45
IKZF3 Q9UKT9 1/20 0.45
PKM P14618 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
HSD17B10 Q99714 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1965253 0.88 CRBN (0.53) CRBNCSNK1A1IKZF2DDB1POLB
SCHEMBL1962505 0.88 CRBN (0.54) CRBNCSNK1A1IKZF2DDB1POLB
SCHEMBL1962494 0.87 CRBN (0.59) CRBNCSNK1A1IKZF2DDB1POLB
SCHEMBL1963650 0.87 CRBN (0.54) CRBNCSNK1A1IKZF2DDB1POLB
SCHEMBL1961641 0.87 ALDH1A1 (0.57) CRBNCSNK1A1IKZF2DDB1POLB
SCHEMBL1961721 0.87 CRBN (0.52) CRBNCSNK1A1IKZF2DDB1POLB
SCHEMBL1962516 0.86 CRBN (0.53) CRBNCSNK1A1IKZF2POLBKDM4E
SCHEMBL1963428 0.86 CRBN (0.62) CRBNCSNK1A1IKZF2DDB1GSPT1
SCHEMBL1962233 0.86 MAPK1 (0.61) CRBNCSNK1A1IKZF2POLBPKM
SCHEMBL1962487 0.86 CRBN (0.52) CRBNCSNK1A1IKZF2DDB1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US claimed
US-20200113896-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY SIGNAL PHARM LLC (US) 2020-04-16 US disclosed
US-20140314752-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY SIGNAL PHARMACEUTICALS, LLC (US) 2014-10-23 US disclosed
EP-1919892-B1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORP (US) 2013-08-14 EP disclosed
US-8481568-B2 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION (US) 2013-07-09 US disclosed
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SEPRACOR INC. 2011-06-16 US disclosed
EP-1919892-A2 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORPORATION (US) 2008-05-14 EP disclosed
WO-2007027527-A2 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORPORATION (US) 2007-03-08 WO disclosed
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200113896-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY MTOR, ULK1, RICTOR CRBN 869/4885CSNK1A1 728/4885IKZF2 401/4885
US-20140314752-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY MTOR, ULK1, RICTOR CRBN 869/4885CSNK1A1 728/4885IKZF2 401/4885
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SI, CYP3A5, CYP2D6 CRBN 2589/4885CSNK1A1 137/4885IKZF2 1965/4885
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same SI, CYP3A5, CYP2D6 CRBN 2589/4885CSNK1A1 137/4885IKZF2 1965/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.